2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists
2-芳基取代的吡啶C区类似物,即2-(3-氟-4-甲基磺酰氨基苯基)丙酰胺,是高效的TRPV1拮抗剂
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2014.05.072
Ryu, HyungChul; Seo, Sejin; Kim, Myeong Seop; Kim, Mi-Yeon; Kim, Ho Shin; Ann, Jihyae; Tran, Phuong-Thao; Hoang, Van-Hai; Byun, Jieun; Cui, Minghua; Son, Karam; Sharma, Pankaz Kumar; Choi, Sun; Blumberg, Peter M; Frank-Foltyn, Robert; Bahrenberg, Gregor; Koegel, Babette-Yvonne; Christoph, Thomas; Frormann, Sven; Lee, Jeewoo