日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sensory neuron-expressed FGF13 controls nociceptive signaling in diabetic neuropathy models

感觉神经元表达的FGF13控制糖尿病神经病变模型中的伤害性信号传导

Singh, Aditya K; Bernabucci, Matteo; Dvorak, Nolan M; Haghighijoo, Zahra; Di Re, Jessica; Goode, Nana A; Kadakia, Feni K; Maile, Laura A; Folorunso, Olumarotimi O; Wadsworth, Paul A; Tapia, Cynthia M; Wang, Pingyuan; Wang, Jigong; Chen, Haiying; Xue, Yu; Singh, Jully; Hankerd, Kali; Gamez, Isaac J; Kager, Makenna; Truong, Vincent; Walsh, Patrick; Shiers, Stephanie I; Kuttanna, Nishka; Liao, Hanyue; Marchi, Margherita; Salvi, Erika; D'Amato, Ilaria; D'Amico, Daniela; Arman, Parsa; Faber, Catharina G; Malik, Rayaz A; de Tommaso, Marina; Ziegler, Dan; Rajarathnam, Krishna; Green, Thomas A; Grace, Peter M; Sapio, Matthew R; Iadarola, Michael J; Cuny, Gregory D; Chow, Diana S; Lauria Pinter, Giuseppe; Davidson, Steve; Green, Dustin P; La, Jun-Ho; Chung, Jin Mo; Zhou, Jia; Price, Theodore J; Salisbury, Elizabeth; Yuan, Subo; Laezza, Fernanda

Inhibition of the GSK3β/Nav1.6 complex suppresses early-stage Alzheimer's hyperexcitability

抑制 GSK3β/Nav1.6 复合物可抑制阿尔茨海默病早期阶段的过度兴奋

Baumgartner, Timothy John; Silva-Pérez, Manuel; Haghighijoo, Zahra; Dvorak, Nolan Michael; Singh, Aditya Kumar; Goode, Nana Aboadwe; Singh, Jully; Grebenkova, Berenice Gutierrez; Marosi, Mate; Di Re, Jessica; Koff, Leandra; Wijitrmektong, Wissarut; Bala, Manu; Liao, Hanyue; Lijffijt, Marijn; Szafran, Adam Thomas; Bolt, Michael James; Mancini, Michael A; Cuny, Gregory D; Chow, Diana Shu-Lian; Limon, Agenor; Chin, Jeannie; Laezza, Fernanda

Role of the Mobile Active Site Flap in IMP Dehydrogenase Inhibitor Binding

移动活性位点瓣在IMP脱氢酶抑制剂结合中的作用

Wang, Xingyou; Rosenberg, Masha M; Kim, Youngchang; Maltseva, Natalia; Cuny, Gregory D; Joachimiak, Andrzej; Kuzmič, Petr; Hedstrom, Lizbeth

Pyridopyrimidinones as a new chemotype of calcium dependent protein kinase 1 (CDPK1) inhibitors for Cryptosporidium

吡啶并嘧啶酮类化合物作为新型钙依赖性蛋白激酶1 (CDPK1) 抑制剂用于治疗隐孢子虫病

Waldron-Young, Elise; Wijitrmektong, Wissarut; Choi, Ryan; Whitman, Grant R; Hulverson, Matthew A; Charania, Raheela; Keelaghan, Aidan; Li, Li; Srinual, Songpol; Nikhar, Sameer; McNamara, Case W; Love, Melissa S; Huerta, Lauren; Bakowski, Malina A; Hu, Ming; Van Voorhis, Wesley C; Mead, Jan R; Cuny, Gregory D

Structure-activity relationship of BMS906024 derivatives for Cryptosporidium parvum growth inhibition

BMS906024衍生物对小隐孢子虫生长抑制的构效关系

Lee, Seungheon; Love, Melissa S; Modukuri, Ramkumar; Chatterjee, Arnab K; Huerta, Lauren; Lawson, Ann P; McNamara, Case W; Mead, Jan R; Hedstrom, Lizbeth; Cuny, Gregory D

Nonhydrolyzable d‑phenylalanine-benzoxazole derivatives retain antitubercular activity

不可水解的D-苯丙氨酸-苯并恶唑衍生物保留抗结核活性

Pepi, Michael J; Chacko, Shibin; Kopetz, Nicole; Boshoff, Helena I M; Cuny, Gregory D; Hedstrom, Lizbeth

An Immunconjugate Vaccine Alters Distribution and Reduces the Antinociceptive, Behavioral and Physiological Effects of Fentanyl in Male and Female Rats

免疫结合疫苗可改变芬太尼在雄性和雌性大鼠体内的分布,并降低芬太尼的镇痛、行为和生理效应。

Haile, Colin N; Baker, Miah D; Sanchez, Sergio A; Lopez Arteaga, Carlos A; Duddupudi, Anantha L; Cuny, Gregory D; Norton, Elizabeth B; Kosten, Thomas R; Kosten, Therese A

Fentanyl conjugate vaccine by injected or mucosal delivery with dmLT or LTA1 adjuvants implicates IgA in protection from drug challenge

芬太尼结合疫苗通过注射或黏膜给药,并辅以dmLT或LTA1佐剂,表明IgA在抵御药物攻击中发挥保护作用。

Stone, Addison E; Scheuermann, Sarah E; Haile, Colin N; Cuny, Gregory D; Velasquez, Marcela Lopez; Linhuber, Joshua P; Duddupudi, Anantha L; Vigliaturo, Jennifer R; Pravetoni, Marco; Kosten, Therese A; Kosten, Thomas R; Norton, Elizabeth B

RIPK protein kinase family: Atypical lives of typical kinases

RIPK蛋白激酶家族:典型激酶的非典型人生

Cuny, Gregory D; Degterev, Alexei

Design of pyrido[2,3-d]pyrimidin-7-one inhibitors of receptor interacting protein kinase-2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling

设计吡啶并[2,3-d]嘧啶-7-酮类受体相互作用蛋白激酶-2 (RIPK2) 和核苷酸结合寡聚化结构域 (NOD) 细胞信号传导抑制剂

Nikhar, Sameer; Siokas, Ioannis; Schlicher, Lisa; Lee, Seungheon; Gyrd-Hansen, Mads; Degterev, Alexei; Cuny, Gregory D