日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Harder than Metal: Challenging Antimicrobial Resistance with Metallo-β-lactamase Inhibitors

比金属更坚硬:用金属β-内酰胺酶抑制剂挑战抗菌素耐药性

De Falco, Antonietta; Alfano, Antonella Ilenia; Cutarella, Luigi; Mori, Mattia; Brindisi, Margherita

Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors.

可持续的 Joullié-Ugi 和连续流实施产生了新型的受卡托普利启发的广谱金属β-内酰胺酶抑制剂

Alfano Antonella Ilenia, Pelliccia Sveva, Barone Simona, Cutarella Luigi, Cancade Sacha Michèle Idriss, Baia Valerio, Cassese Emilia, Russomanno Pasquale, Messano Nicolò, Frank Denia, Weizel Lilia, Rotter Marco J, Brunst Steffen, Wichelhaus Thomas A, Proschak Ewgenij, Tedesco Daniele, Mori Mattia, Docquier Jean Denis, Summa Vincenzo, Brindisi Margherita

Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus

他莫昔芬衍生物对耐甲氧西林金黄色葡萄球菌的抗菌活性

Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S; Smani, Younes

Retargeting Gram-Positive-Only Adarotene-Derived Antibacterials to Broad-Spectrum Antibiotics

将仅针对革兰氏阳性菌的阿达罗汀衍生物抗菌药物重新定位为广谱抗生素

Princiotto, Salvatore; Cutarella, Luigi; Fortuna, Alessandra; Mellini, Marta; Casciaro, Bruno; Loffredo, Maria Rosa; Temprano, Alvaro G; Cappiello, Floriana; Leoni, Livia; Mangoni, Maria Luisa; Mori, Mattia; Musso, Loana; Sacchi, Francesca; Pinna, Cecilia; Rampioni, Giordano; Dallavalle, Sabrina; Pisano, Claudio

Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid

基于香豆酸的新型人碳酸酐酶抑制剂的设计、合成、分子建模研究和生物学研究

Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T

The Antiepileptic Drug Levetiracetam Inhibits Carbonic Anhydrase: In Vitro and In Silico Studies on Catalytically Active Human Isoforms

抗癫痫药物左乙拉西坦抑制碳酸酐酶:对具有催化活性的人类同工酶的体外和计算机模拟研究

Cutarella, Luigi; Mori, Mattia; Supuran, Claudiu T

Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors

新型2,4-二氯-5-氨磺酰基苯甲酸肟酯:作为潜在的人类碳酸酐酶抑制剂的初步研究

Kilbile, Jaydeo T; Sapkal, Suryakant B; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T