Triazole 187 is a biased KOR agonist that suppresses itch without sedation and induces anxiolytic-like behaviors in mice
三唑187是一种偏向性κ阿片受体激动剂,可在不引起镇静的情况下抑制瘙痒,并诱导小鼠产生类似抗焦虑的行为。
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影响因子:
doi:10.1101/2025.02.17.638680
Volf, Allison; Brust, Tarsis F; Kobylski, Robin R; Czekner, Kerri M; Stahl, Edward L; Cameron, Michael D; Trojniak, Ashley E; Aubé, Jeffrey; Bohn, Laura M