日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting phosphatases in cancer: suppression of many versus the ablation of one

癌症治疗中靶向磷酸酶:抑制多种磷酸酶与仅消除一种磷酸酶。

D'Arcy, Brandon M; Prakash, Aishwarya; Honkanen, Richard E

PP1:Tautomycetin Complex Reveals a Path toward the Development of PP1-Specific Inhibitors

PP1:tautomycetin复合物揭示了开发PP1特异性抑制剂的途径

Choy, Meng S; Swingle, Mark; D'Arcy, Brandon; Abney, Kevin; Rusin, Scott F; Kettenbach, Arminja N; Page, Rebecca; Honkanen, Richard E; Peti, Wolfgang

An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C)

丝氨酸/苏氨酸蛋白磷酸酶1型和5型(PP1C和PP5C)催化抑制剂的超高通量筛选

Swingle, Mark; Volmar, Claude-Henry; Saldanha, S Adrian; Chase, Peter; Eberhart, Christina; Salter, Edward A; D'Arcy, Brandon; Schroeder, Chad E; Golden, Jennifer E; Wierzbicki, Andrzej; Hodder, Peter; Honkanen, Richard E

Crystal structures and mutagenesis of PPP-family ser/thr protein phosphatases elucidate the selectivity of cantharidin and novel norcantharidin-based inhibitors of PP5C.

PPP家族丝氨酸/苏氨酸蛋白磷酸酶的晶体结构和诱变研究阐明了斑蝥素和新型去甲斑蝥素类PP5C抑制剂的选择性

Chattopadhyay Debasish, Swingle Mark R, Salter Edward A, Wood Eric, D'Arcy Brandon, Zivanov Catherine, Abney Kevin, Musiyenko Alla, Rusin Scott F, Kettenbach Arminja, Yet Larry, Schroeder Chad E, Golden Jennifer E, Dunham Wade H, Gingras Anne-Claude, Banerjee Surajit, Forbes David, Wierzbicki Andrzej, Honkanen Richard E