日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tracking the cellular uptake and phototoxicity of Ru(ii)-polypyridyl-1,8-naphthalimide Tröger's base conjugates

追踪 Ru(ii)-聚吡啶-1,8-萘酰亚胺 Tröger 碱缀合物的细胞摄取和光毒性

Bright, Sandra A; Erby, MariaLuisa; Poynton, Fergus E; Monteyne, Daniel; Pérez-Morga, David; Gunnlaugsson, Thorfinnur; Williams, D Clive; Elmes, Robert B P

Synthesis and Biochemical Evaluation of Ethanoanthracenes and Related Compounds: Antiproliferative and Pro-Apoptotic Effects in Chronic Lymphocytic Leukemia (CLL)

乙基蒽和相关化合物的合成和生化评价:在慢性淋巴细胞白血病 (CLL) 中的抗增殖和促凋亡作用

James P McKeown, Andrew J Byrne, Sandra A Bright, Clara E Charleton, Shubhangi Kandwal, Ivan Čmelo, Brendan Twamley, Anthony M McElligott, Darren Fayne, Niamh M O'Boyle, D Clive Williams, Mary J Meegan

Synthesis and Pro-Apoptotic Effects of Nitrovinylanthracenes and Related Compounds in Chronic Lymphocytic Leukaemia (CLL) and Burkitt's Lymphoma (BL)

硝基乙烯基蒽及其相关化合物在慢性淋巴细胞白血病 (CLL) 和伯基特淋巴瘤 (BL) 中的合成及其促凋亡作用

Andrew J Byrne, Sandra A Bright, James P McKeown, Adam Bergin, Brendan Twamley, Anthony M McElligott, Sara Noorani, Shubhangi Kandwal, Darren Fayne, Niamh M O'Boyle, D Clive Williams, Mary J Meegan

Design, Synthesis and Biochemical Evaluation of Novel Ethanoanthracenes and Related Compounds to Target Burkitt's Lymphoma

针对伯基特淋巴瘤的新型乙蒽及相关化合物的设计、合成和生化评估

Andrew J Byrne, Sandra A Bright, James P McKeown, John E O'Brien, Brendan Twamley, Darren Fayne, D Clive Williams, Mary J Meegan

The pyrrolo-1,5-benzoxazepine, PBOX-15, enhances TRAIL‑induced apoptosis by upregulation of DR5 and downregulation of core cell survival proteins in acute lymphoblastic leukaemia cells

吡咯并-1,5-苯并恶唑并化合物PBOX-15通过上调DR5和下调急性淋巴细胞白血病细胞中核心细胞存活蛋白的表达,增强TRAIL诱导的细胞凋亡。

Nathwani, Seema-Maria; Greene, Lisa M; Butini, Stefania; Campiani, Giuseppe; Williams, D Clive; Samali, Afshin; Szegezdi, Eva; Zisterer, Daniela M

Antitumor effect of pyrrolo-1,5-benzoxazepine-15 and its synergistic effect with Oxaliplatin and 5-FU in colorectal cancer cells

吡咯并-1,5-苯并氧氮卓-15对结直肠癌细胞的抗肿瘤作用及其与奥沙利铂和5-FU的协同作用

Donatella Fiore, Maria Chiara Proto, Simona Pisanti, Paola Picardi, Antonio Christian Pagano Zottola, Stefania Butini, Sandra Gemma, Alice Casagni, Chiara Laezza, Mario Vitale, Alessia Ligresti, Vincenzo Di Marzo, Daniela M Zisterer, Seema Nathwani, D Clive Williams, Giuseppe Campiani, Patrizia Gazz

"True" antiandrogens-selective non-ligand-binding pocket disruptors of androgen receptor-coactivator interactions: novel tools for prostate cancer

“真正的”抗雄激素选择性非配体结合口袋干扰剂,可破坏雄激素受体-辅激活因子相互作用:治疗前列腺癌的新工具

Laura Caboni, Gemma K Kinsella, Fernando Blanco, Darren Fayne, William N Jagoe, Miriam Carr, D Clive Williams, Mary J Meegan, David G Lloyd

Pyrrolo-1,5-Benzoxazepines Induce Apoptosis in Chronic Myeloid Leukemia (CML) Cells by Bypassing the Apoptotic Suppressor BCR-ABL

吡咯并-1,5-苯并恶唑类化合物通过绕过凋亡抑制因子BCR-ABL诱导慢性粒细胞白血病(CML)细胞凋亡。

Mc Gee, Margaret M; Campiani, Giuseppe; Ramunno, Anna; Fattorusso, Caterina; Nacci, Vito; Lawler, Mark; Williams, D Clive; Zisterer, Daniela M