日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A mild and atom-efficient four-component cascade strategy for the construction of biologically relevant 4-hydroxyquinolin-2(1H)-one derivatives

一种温和且原子经济的四组分级联策略,用于构建具有生物学意义的4-羟基喹啉-2(1H)-酮衍生物

Grishin, Dmitrii A; Sharkovskaia, Kseniia I; Kolmakov, Ilya G; Ipatova, Daria A; Petrov, Rostislav A; Dagaev, Nikolai D; Skvortsov, Dmitry A; Khrenova, Maria G; Andreychev, Valeriy V; Evteev, Sergei A; Ivanenkov, Yan A; Antipin, Roman L; Dontsova, Olga А; Beloglazkina, Elena K

Design, Synthesis, and Biological Evaluation of 6″-Modified Apramycin Derivatives to Overcome Aminoglycoside Resistance

设计、合成及生物学评价6″-修饰的阿普拉霉素衍生物以克服氨基糖苷类耐药性

Shapovalova, Kseniya S; Zatonsky, Georgy V; Razumova, Elizaveta A; Dagaev, Nikolai D; Lukianov, Dmitrii A; Grammatikova, Natalia E; Tikhomirov, Alexander S; Shchekotikhin, Andrey E

Characterization of Bacillus velezensis EV17 and K-3618 and Their Polyketide Antibiotic Oxydifficidin, an Inhibitor of Prokaryotic Translation with Low Cytotoxicity

贝莱斯芽孢杆菌EV17和K-3618的特性及其聚酮类抗生素Oxydifficidin(一种低细胞毒性的原核翻译抑制剂)

Chernyshova, Alisa P; Marina, Valeriya I; Tereshchenkov, Andrey G; Sagitova, Vladislava E; Kryakvin, Maksim A; Dagaev, Nikolai D; Yurchenko, Eugeniya G; Arzamazova, Kseniya A; Guglya, Elena B; Belozerova, Olga A; Kovalchuk, Sergey I; Baranova, Margarita N; Kudzhaev, Arsen M; Shikov, Anton E; Romanenko, Maria N; Rudenko, Alexander Yu; Chebotar, Vladimir K; Gancheva, Maria S; Baganova, Maria E; Biryukov, Mikhail V; Panova, Tatiana V; Khrenova, Maria G; Tashlitsky, Vadim N; Sumbatyan, Natalia V; Zakalyukina, Yulia V; Antonets, Kirill S; Nizhnikov, Anton A; Polshakov, Vladimir I; Terekhov, Stanislav S; Zvereva, Maria I; Dontsova, Olga A; Sergiev, Petr V; Alferova, Vera A; Lukianov, Dmitrii A

Synthesis and Biological Evaluation of Benzo [4,5]- and Naphtho[2',1':4,5]imidazo[1,2-c]pyrimidinone Derivatives

苯并[4,5]-和萘并[2',1':4,5]咪唑并[1,2-c]嘧啶酮衍生物的合成及生物学评价

Kamzeeva, Polina; Dagaev, Nikolai; Lizunova, Sofia; Khodarovich, Yuri; Sogomonyan, Anna; Kolchanova, Anastasia; Pokrovsky, Vadim; Alferova, Vera; Chistov, Alexey; Eshtukov-Shcheglov, Artur; Eshtukova-Shcheglova, Elizaveta; Belyaev, Evgeny; Skvortsov, Dmitry; Varizhuk, Anna; Aralov, Andrey