日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Late-stage peptide modification with salicylaldehyde tag enhances affinity for nuclear factor-kappa B essential modulator

后期肽修饰用水杨醛标签增强了对核因子-κB必需调节剂的亲和力

Mason, Mattia; Peqini, Kaliroi; Uggeri, Federico; Rondelli, Diego; Sattin, Sara; Pignataro, Luca; Pellegrino, Sara; Belvisi, Laura; Scarpa, Edoardo; Bucci, Raffaella; Dal Corso, Alberto

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker

利用体外质谱法对带有蛋白酶可切割和酸不稳定连接子的抗体-瑞喹莫德偶联物进行生物分布分析

Bisbal Lopez, Lydia; Ravazza, Domenico; Bocci, Matilde; Zana, Aureliano; Principi, Lucrezia; Dakhel Plaza, Sheila; Galbiati, Andrea; Gilardoni, Ettore; Scheuermann, Jörg; Neri, Dario; Pignataro, Luca; Gennari, Cesare; Cazzamalli, Samuele; Dal Corso, Alberto

Visible Light-Promoted β-Functionalization of Carbonyl Compounds in the Presence of Organic Dyes

可见光促进有机染料存在下羰基化合物的β-官能化

Dolcini, Luigi; Gandini, Tommaso; Castiglioni, Riccardo; Bossi, Alberto; Penconi, Marta; Dal Corso, Alberto; Gennari, Cesare; Pignataro, Luca

Advanced Pyrrolidine-Carbamate Self-Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release

具有叔胺基团的先进吡咯烷-氨基甲酸酯自毁间隔基可诱导超快速循环药物释放

Dal Corso, Alberto; Frigoli, Margaux; Prevosti, Martina; Mason, Mattia; Bucci, Raffaella; Belvisi, Laura; Pignataro, Luca; Gennari, Cesare

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

中性粒细胞弹性蛋白酶促进连接子裂解和紫杉醇从整合素靶向缀合物中释放

Raposo Moreira Dias, André; Pina, Arianna; Dean, Amelia; Lerchen, Hans-Georg; Caruso, Michele; Gasparri, Fabio; Fraietta, Ivan; Troiani, Sonia; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α(V) β(3)

靶向整合素α(V)β(3)的RGD和isoDGR-单甲基奥瑞他汀缀合物的合成和生物学评价

Raposo Moreira Dias, André; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkühler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto

Protease-Cleavable Linkers Modulate the Anticancer Activity of Noninternalizing Antibody-Drug Conjugates

蛋白酶可切割连接子调节非内吞抗体-药物偶联物的抗癌活性

Dal Corso, Alberto; Cazzamalli, Samuele; Gébleux, Rémy; Mattarella, Martin; Neri, Dario

Acetazolamide Serves as Selective Delivery Vehicle for Dipeptide-Linked Drugs to Renal Cell Carcinoma

乙酰唑胺作为二肽连接药物选择性递送载体,靶向肾细胞癌

Cazzamalli, Samuele; Dal Corso, Alberto; Neri, Dario

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors.

靶向αvβ3整合素和VEGF受体的双作用配体的合成、表征和生物学评价

Zanella Simone, Mingozzi Michele, Dal Corso Alberto, Fanelli Roberto, Arosio Daniela, Cosentino Marco, Schembri Laura, Marino Franca, De Zotti Marta, Formaggio Fernando, Pignataro Luca, Belvisi Laura, Piarulli Umberto, Gennari Cesare