日期 影响因子
日期:
2020 年 — 2026 年
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影响因子:
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Discovery of Axelopran (TD-1211): A Peripherally Restricted μ-Opioid Receptor Antagonist

Axelopran (TD-1211) 的发现：一种外周限制性 μ-阿片受体拮抗剂

期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.9b00406
Long, Daniel D; Armstrong, Scott R; Beattie, David T; Campbell, Christina B; Church, Timothy J; Colson, Pierre-Jean; Dalziel, Sean M; Jacobsen, John R; Jiang, Lan; Obedencio, Glenmar P; Rapta, Miroslav; Saito, Daisuke; Stergiades, Ioanna; Tsuruda, Pamela R; Van Dyke, Priscilla M; Vickery, Ross G
信号转导
发表日期：2019
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Development and binding mode assessment of N-[4-[2-propyn-1-yl[(6S)-4,6,7,8-tetrahydro-2-(hydroxymethyl)-4-oxo-3H-cyclopenta[g]quinazolin-6-yl]amino]benzoyl]-l-γ-glutamyl-D-glutamic acid (BGC 945), a novel thymidylate synthase inhibitor that targets tumor cells.

对靶向肿瘤细胞的新型胸苷酸合成酶抑制剂 N-[4-[2-丙炔-1-基[(6S)-4,6,7,8-四氢-2-(羟甲基)-4-氧代-3H-环戊并[g]喹唑啉-6-基]氨基]苯甲酰基]-l-γ-谷氨酰-D-谷氨酸 (BGC 945) 进行开发和结合模式评估

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm400490e
Tochowicz Anna, Dalziel Sean, Eidam Oliv, O'Connell Joseph D 3rd, Griner Sarah, Finer-Moore Janet S, Stroud Robert M
肿瘤
发表日期：2013
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