Discovery of 2-amide-3-methylester thiophenes that target SARS-CoV-2 Mac1 and repress coronavirus replication, validating Mac1 as an anti-viral target
发现 2-酰胺-3-甲酯噻吩类化合物,该化合物可靶向 SARS-CoV-2 Mac1 并抑制冠状病毒复制,从而证实 Mac1 可作为抗病毒靶点
期刊:
影响因子:
doi:10.1101/2023.08.28.555062
Sarah Wazir, Tomi A O Parviainen, Jessica J Pfannenstiel, Men Thi Hoai Duong, Daniel Cluff, Sven T Sowa, Albert Galera-Prat, Dana Ferraris, Mirko M Maksimainen, Anthony R Fehr, Juha P Heiskanen, Lari Lehtiö