日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulation of succinyl-CoA:3-ketoacid CoA transferase activity by a single amino acid residue in acetate:succinate CoA transferase from Trypanosoma brucei, the causative agent of African sleeping sickness

锥虫(非洲昏睡病病原体)乙酸:琥珀酸CoA转移酶中单个氨基酸残基对琥珀酰CoA:3-酮酸CoA转移酶活性的调节

Mochizuki, Kota; Inaoka, Daniel Ken; Fukuda, Keisuke; Kurasawa, Hana; Iyoda, Kenji; Nakai, Uta; Harada, Shigeharu; Balogun, Emmanuel O; Bringaud, Frédéric; Boshart, Michael; Sakura, Takaya; Hirayama, Kenji; Kita, Kiyoshi; Shiba, Tomoo

Pivotal roles of Plasmodium falciparum lysophospholipid acyltransferase 1 in cell cycle progression and cytostome internalization

恶性疟原虫溶血磷脂酰基转移酶1在细胞周期进程和胞口内吞作用中的关键作用

Junpei Fukumoto,Minako Yoshida #,Suzumi M Tokuoka #,Eri Saki H Hayakawa #,Shinya Miyazaki,Takaya Sakura,Daniel Ken Inaoka,Kiyoshi Kita,Jiro Usukura,Hideo Shindou,Fuyuki Tokumasu

Development of tolerance to bedaquiline by overexpression of trypanosomal acetate: succinate CoA transferase in Mycobacterium smegmatis

耻垢分枝杆菌中锥虫乙酸:琥珀酸CoA转移酶过表达导致对贝达喹啉产生耐受性

Gloria Mavinga Bundutidi,Kota Mochizuki,Yuichi Matsuo,Mizuki Hayashishita,Takaya Sakura,Yuri Ando,Gregory Murray Cook,Acharjee Rajib,Frédéric Bringaud,Michael Boshart,Shinjiro Hamano,Masakazu Sekijima,Kenji Hirayama,Kiyoshi Kita,Daniel Ken Inaoka

Accelerating Antimalarial Drug Discovery with a New High-Throughput Screen for Fast-Killing Compounds

利用新型高通量筛选快速杀灭化合物加速抗疟药物发现

Sakura, Takaya; Ishii, Ryuta; Yoshida, Eri; Kita, Kiyoshi; Kato, Teruhisa; Inaoka, Daniel Ken

A versatile Plasmodium falciparum reporter line expressing NanoLuc enables highly sensitive multi-stage drug assays

表达 NanoLuc 的多功能恶性疟原虫报告系可实现高灵敏度的多阶段药物检测

Yukiko Miyazaki, Martijn W Vos, Fiona J A Geurten, Pierre Bigeard, Hans Kroeze, Shohei Yoshioka, Mitsuhiro Arisawa, Daniel Ken Inaoka, Valerie Soulard, Koen J Dechering, Blandine Franke-Fayard, Shinya Miyazaki

Fumarate respiration of Fasciola flukes as a potential drug target

以肝片吸虫的富马酸呼吸作用作为潜在药物靶点

Tashibu, Atsushi; Inaoka, Daniel Ken; Sakamoto, Kimitoshi; Murakami, Kenji; Zannatul, Ferdoush; Kita, Kiyoshi; Ichikawa-Seki, Madoka

Killing Two Birds with One Stone: Discovery of Dual Inhibitors of Oxygen and Fumarate Respiration in Zoonotic Parasite, Echinococcus multilocularis

一石二鸟:在人畜共患寄生虫多房棘球绦虫中发现氧气和富马酸呼吸的双重抑制剂

Enkai, Shigehiro; Kouguchi, Hirokazu; Inaoka, Daniel Ken; Shiba, Tomoo; Hidaka, Masahito; Matsuyama, Hiroyuki; Sakura, Takaya; Yagi, Kinpei; Kita, Kiyoshi

Discovery of a Hidden Trypanosoma cruzi Spermidine Synthase Binding Site and Inhibitors through In Silico, In Vitro, and X-ray Crystallography

通过计算机模拟、体外实验和X射线晶体学方法发现克氏锥虫亚精胺合酶的隐藏结合位点及其抑制剂

Yoshino, Ryunosuke; Yasuo, Nobuaki; Hagiwara, Yohsuke; Ishida, Takashi; Inaoka, Daniel Ken; Amano, Yasushi; Tateishi, Yukihiro; Ohno, Kazuki; Namatame, Ichiji; Niimi, Tatsuya; Orita, Masaya; Kita, Kiyoshi; Akiyama, Yutaka; Sekijima, Masakazu

Biochemical characterization and identification of ferulenol and embelin as potent inhibitors of malate:quinone oxidoreductase from Campylobacter jejuni

对空肠弯曲菌中苹果酸:醌氧化还原酶的强效抑制剂ferulenol和embelin进行生化表征和鉴定

Kabongo, Augustin Tshibaka; Acharjee, Rajib; Sakura, Takaya; Bundutidi, Gloria Mavinga; Hartuti, Endah Dwi; Davies, Cadi; Gundogdu, Ozan; Kita, Kiyoshi; Shiba, Tomoo; Inaoka, Daniel Ken

Antiviral activity of 5-aminolevulinic acid against variants of severe acute respiratory syndrome coronavirus 2

5-氨基乙酰丙酸对严重急性呼吸综合征冠状病毒2变异株的抗病毒活性

Ngwe Tun, Mya Myat; Sakura, Takaya; Sakurai, Yasuteru; Kurosaki, Yohei; Inaoka, Daniel Ken; Shioda, Norifumi; Yasuda, Jiro; Kita, Kiyoshi; Morita, Kouichi