Preclinical anti-myeloma activity of EDO-S101, a new bendamustine-derived molecule with added HDACi activity, through potent DNA damage induction and impairment of DNA repair
EDO-S101 是一种新型苯达莫司汀衍生分子,具有附加的 HDACi 活性,可通过强效诱导 DNA 损伤和破坏 DNA 修复,发挥临床前抗骨髓瘤活性
期刊:Journal of Hematology & Oncology
影响因子:29.5
doi:10.1186/s13045-017-0495-y
Ana-Alicia López-Iglesias, Ana B Herrero, Marta Chesi, Laura San-Segundo, Lorena González-Méndez, Susana Hernández-García, Irena Misiewicz-Krzeminska, Dalia Quwaider, Montserrat Martín-Sánchez, Daniel Primo, Teresa Paíno, P Leif Bergsagel, Thomas Mehrling, Marcos González-Díaz, Jesús F San-Miguel, M