日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Privileged Scaffold Hybridization in the Design of Carbonic Anhydrase Inhibitors

碳酸酐酶抑制剂设计中的特权支架杂交

Daniela Secci, Erica Sanna, Simona Distinto, Alessia Onali, Antonio Lupia, Laura Demuru, Giulia Atzeni, Rita Meleddu, Filippo Cottiglia, Andrea Angeli, Claudiu T Supuran, Elias Maccioni

Inhibition of intestinal inflammation and fibrosis by Scutellaria Baicalensis georgi and Boswellia serrata in human epithelial cells and fibroblasts

黄芩和乳香树对人类上皮细胞和成纤维细胞中肠道炎症和纤维化的抑制作用

Ilaria Laudadio, Beatrice Leter, Francesca Palone, Salvatore Cucchiara, Claudia Carissimi, Noemi Scafa, Daniela Secci, Roberta Vitali, Laura Stronati

Chiral Hydroxy Metabolite of Mebendazole: Analytical and Semi-Preparative High-Performance Liquid Chromatography Resolution and Chiroptical Properties

甲苯咪唑手性羟基代谢物:分析和半制备高效液相色谱分离和手性光学性质

Paolo Guglielmi, Gaia Pulitelli, Francesca Arrighi, Daniela Secci, Marco Pierini, Roberto Cirilli

Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa

发现并优化基于苯并噻唑支架的 DNA 旋转酶抑制剂,该抑制剂对鲍曼不动杆菌和铜绿假单胞菌具有强效活性

Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Pa

A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration

对抗神经炎症的多靶点方法:烷基取代的香豆素作为神经退行性疾病相关酶的抑制剂

Emanuela Berrino, Simone Carradori, Fabrizio Carta, Francesco Melfi, Marialucia Gallorini, Giulio Poli, Tiziano Tuccinardi, José G Fernández-Bolaños, Óscar López, Jacobus P Petzer, Anél Petzer, Paolo Guglielmi, Daniela Secci, Claudiu T Supuran

Inhibition of lysine acetyltransferases impairs tumor angiogenesis acting on both endothelial and tumor cells

抑制赖氨酸乙酰转移酶可损害作用于内皮细胞和肿瘤细胞的肿瘤血管生成

Marta Di Martile, Chiara Gabellini, Marianna Desideri, Marta Matraxia, Valentina Farini, Elisabetta Valentini, Simone Carradori, Cristiana Ercolani, Simonetta Buglioni, Daniela Secci, Massimiliano Andreazzoli, Donatella Del Bufalo, Daniela Trisciuoglio

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

开放糖精基二级磺胺类药物作为癌症相关碳酸酐酶 IX 和 XII 异构体的强效和选择性抑制剂

Melissa D'Ascenzio, Paolo Guglielmi, Simone Carradori, Daniela Secci, Rosalba Florio, Adriano Mollica, Mariangela Ceruso, Atilla Akdemir, Anatoly P Sobolev, Claudiu T Supuran

Histone acetyltransferase inhibitor CPTH6 preferentially targets lung cancer stem-like cells

组蛋白乙酰转移酶抑制剂 CPTH6 优先靶向肺癌干细胞

Marta Di Martile, Marianna Desideri, Teresa De Luca, Chiara Gabellini, Simonetta Buglioni, Adriana Eramo, Giovanni Sette, Michele Milella, Dante Rotili, Antonello Mai, Simone Carradori, Daniela Secci, Ruggero De Maria, Donatella Del Bufalo, Daniela Trisciuoglio

CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells

噻唑衍生物 CPTH6 诱导人类白血病细胞组蛋白低乙酰化和凋亡

Daniela Trisciuoglio, Ylenia Ragazzoni, Andrea Pelosi, Marianna Desideri, Simone Carradori, Chiara Gabellini, Giovanna Maresca, Riccardo Nescatelli, Daniela Secci, Adriana Bolasco, Bruna Bizzarri, Chiara Cavaliere, Igea D'Agnano, Patrizia Filetici, Lucia Ricci-Vitiani, Maria Giulia Rizzo, Donatella