日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Simultaneous Combination of the CDK4/6 Inhibitor Palbociclib With Regorafenib Induces Enhanced Anti-tumor Effects in Hepatocarcinoma Cell Lines

CDK4/6 抑制剂 Palbociclib 与瑞戈非尼同时联合使用可在肝癌细胞系中增强抗肿瘤作用

Graziana Digiacomo, Claudia Fumarola, Silvia La Monica, Mara A Bonelli, Daniele Cretella, Roberta Alfieri, Andrea Cavazzoni, Maricla Galetti, Patrizia Bertolini, Gabriele Missale, Pier Giorgio Petronini

Pemetrexed Enhances Membrane PD-L1 Expression and Potentiates T Cell-Mediated Cytotoxicity by Anti-PD-L1 Antibody Therapy in Non-Small-Cell Lung Cancer

培美曲塞通过抗 PD-L1 抗体疗法增强非小细胞肺癌中的膜 PD-L1 表达并增强 T 细胞介导的细胞毒性

Andrea Cavazzoni, Graziana Digiacomo, Roberta Alfieri, Silvia La Monica, Claudia Fumarola, Maricla Galetti, Mara Bonelli, Daniele Cretella, Valeria Barili, Alessandra Zecca, Elisa Giovannetti, Michelangelo Fiorentino, Marcello Tiseo, Pier Giorgio Petronini, Andrea Ardizzoni

Pre-treatment with the CDK4/6 inhibitor palbociclib improves the efficacy of paclitaxel in TNBC cells

使用 CDK4/6 抑制剂 palbociclib 进行预处理可提高紫杉醇对 TNBC 细胞的疗效

Daniele Cretella, Claudia Fumarola, Mara Bonelli, Roberta Alfieri, Silvia La Monica, Graziana Digiacomo, Andrea Cavazzoni, Maricla Galetti, Daniele Generali, Pier Giorgio Petronini

Expanding the Arsenal of FGFR Inhibitors: A Novel Chloroacetamide Derivative as a New Irreversible Agent With Anti-proliferative Activity Against FGFR1-Amplified Lung Cancer Cell Lines

扩大 FGFR 抑制剂库:一种新型氯乙酰胺衍生物作为新型不可逆药物,对 FGFR1 扩增肺癌细胞系具有抗增殖活性

Claudia Fumarola, Nicole Bozza, Riccardo Castelli, Francesca Ferlenghi, Giuseppe Marseglia, Alessio Lodola, Mara Bonelli, Silvia La Monica, Daniele Cretella, Roberta Alfieri, Roberta Minari, Maricla Galetti, Marcello Tiseo, Andrea Ardizzoni, Marco Mor, Pier Giorgio Petronini

The anti-tumor efficacy of CDK4/6 inhibition is enhanced by the combination with PI3K/AKT/mTOR inhibitors through impairment of glucose metabolism in TNBC cells

CDK4/6 抑制剂与 PI3K/AKT/mTOR 抑制剂联合使用可增强其抗肿瘤功效,因为该抑制剂可损害 TNBC 细胞中的葡萄糖代谢

Daniele Cretella, Andrea Ravelli, Claudia Fumarola, Silvia La Monica, Graziana Digiacomo, Andrea Cavazzoni, Roberta Alfieri, Alessandra Biondi, Daniele Generali, Mara Bonelli, Pier Giorgio Petronini

Enhanced efficacy of AKT and FAK kinase combined inhibition in squamous cell lung carcinomas with stable reduction in PTEN

AKT 和 FAK 激酶联合抑制对鳞状细胞肺癌的疗效增强,PTEN 稳定降低

Andrea Cavazzoni, Silvia La Monica, Roberta Alfieri, Andrea Ravelli, Nele Van Der Steen, Rocco Sciarrillo, Denise Madeddu, Costanza Anna Maria Lagrasta, Federico Quaini, Mara Bonelli, Claudia Fumarola, Daniele Cretella, Graziana Digiacomo, Marcello Tiseo, Godefridus J Peters, Andrea Ardizzoni, Pier

Effect of ABCG2/BCRP Expression on Efflux and Uptake of Gefitinib in NSCLC Cell Lines

ABCG2/BCRP 表达对 NSCLC 细胞系中吉非替尼流出和吸收的影响

Maricla Galetti, Pier Giorgio Petronini, Claudia Fumarola, Daniele Cretella, Silvia La Monica, Mara Bonelli, Andrea Cavazzoni, Francesca Saccani, Cristina Caffarra, Roberta Andreoli, Antonio Mutti, Marcello Tiseo, Andrea Ardizzoni, Roberta R Alfieri