日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and Characterization of a First-in-Class LIV1-TLR7/8 Immunomodulatory Conjugate with Robust Myeloid Activation and Antitumor Activity.

发现并表征了具有强大髓系激活和抗肿瘤活性的首创 LIV1-TLR7/8 免疫调节偶联物

Yamazoe Sayumi, Poudel Yam, Sega Emanuela, Mukhopadhyay Anandaroop, Ramakrishnan Radha, Ukairo Okechukwu, Liu Scot, Akter Rahima, Sadanala Keerthi, Que Kathryn, Cheng Qinqin, Kotapati Srikanth, Deshpande Madhura, Cox Matthew, Chourey Shishir, Gupta Anuradha, Kempson James, Pabbisetty Kumar, Kaspady Mahammed, Bhattasali Debabrata, Yip Shiuhang, Wu Dauh-Rurng, Pookot Deepa, Li Yvonne, Kozhich Alexander, Drexler Dieter, Carl Stephen, Deyanova Ekaterina, Smith Michael, Chan Henry, West Sean, Diong S J, Chang Aram, Florin Lore, Mathur Arvind, Strop Pavel, Zapf Christoph W, Law Deborah, Wilson Nicholas, Broz Miranda, Chekler Eugene P

Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist

BMS-986251 的发现:一种临床上可行、高效且选择性的 RORγt 反向激动剂

Cherney, Robert J; Cornelius, Lyndon A M; Srivastava, Anurag; Weigelt, Carolyn A; Marcoux, David; Duan, James J-W; Shi, Qing; Batt, Douglas G; Liu, Qingjie; Yip, Shiuhang; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John; Khan, Javed; Wang, Jinhong; Yarde, Melissa; Cvijic, Mary Ellen; Mathur, Arvind; Li, Sha; Shuster, David; Khandelwal, Purnima; Borowski, Virna; Xie, Jenny; Obermeier, Mary; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Tino, Joseph A; Macor, John E; Salter-Cid, Luisa; Denton, Rex; Zhao, Qihong; Carter, Percy H; Dhar, T G Murali

Driving Potency with Rotationally Stable Atropisomers: Discovery of Pyridopyrimidinedione-Carbazole Inhibitors of BTK

利用旋转稳定的阻转异构体增强效力:发现吡啶并嘧啶二酮-咔唑类BTK抑制剂

Srivastava, Anurag S; Ko, Soo; Watterson, Scott H; Pattoli, Mark A; Skala, Stacey; Cheng, Lihong; Obermeier, Mary T; Vickery, Rodney; Discenza, Lorell N; D'Arienzo, Celia J; Gillooly, Kathleen M; Taylor, Tracy L; Pulicicchio, Claudine; McIntyre, Kim W; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Dai, Jun; Wang, Chunlei; Zhang, Yingru; Wang, Bei; Pawluczyk, Joseph; Kempson, James; Zhao, Rulin; Hou, Xiaoping; Rampulla, Richard; Mathur, Arvind; Galella, Michael A; Salter-Cid, Luisa; Barrish, Joel C; Carter, Percy H; Fura, Aberra; Burke, James R; Tino, Joseph A

Identification of potent tricyclic prodrug S1P(1) receptor modulators

鉴定强效三环类前药S1P(1)受体调节剂

Marcoux, David; Xiao, Hai-Yun; Murali Dhar, T G; Xie, Jenny; Lehman-McKeeman, Lois D; Wu, Dauh-Rurng; Dabros, Marta; Yang, Xiaoxia; Taylor, Tracy L; Zhou, Xia D; Heimrich, Elizabeth M; Thomas, Rochelle; McIntyre, Kim W; Shi, Hong; Levesque, Paul C; Sun, Huadong; Yang, Zheng; Marino, Anthony M; Cornelius, Georgia; D'Arienzo, Celia J; Gupta, Anuradha; Pragalathan, Bala; Rampulla, Richard; Mathur, Arvind; Shen, Ding Ren; Cvijic, Mary Ellen; Salter-Cid, Luisa; Lombardo, Louis J; Carter, Percy H; Dyckman, Alaric J

Identification and Preclinical Pharmacology of BMS-986104: A Differentiated S1P1 Receptor Modulator in Clinical Trials

BMS-986104的鉴定和临床前药理学研究:一种在临床试验中应用的差异化S1P1受体调节剂

Dhar, T G Murali; Xiao, Hai-Yun; Xie, Jenny; Lehman-McKeeman, Lois D; Wu, Dauh-Rurng; Dabros, Marta; Yang, Xiaoxia; Taylor, Tracy L; Zhou, Xia D; Heimrich, Elizabeth M; Thomas, Rochelle; McIntyre, Kim W; Warrack, Bethanne; Shi, Hong; Levesque, Paul C; Zhu, Jia L; Hennan, James; Balimane, Praveen; Yang, Zheng; Marino, Anthony M; Cornelius, Georgia; D'Arienzo, Celia J; Mathur, Arvind; Shen, Ding Ren; Cvijic, Mary Ellen; Salter-Cid, Luisa; Barrish, Joel C; Carter, Percy H; Dyckman, Alaric J

Discovery of Clinical Candidate BMS-906024: A Potent Pan-Notch Inhibitor for the Treatment of Leukemia and Solid Tumors

临床候选药物BMS-906024的发现:一种用于治疗白血病和实体瘤的强效泛Notch抑制剂

Gavai, Ashvinikumar V; Quesnelle, Claude; Norris, Derek; Han, Wen-Ching; Gill, Patrice; Shan, Weifang; Balog, Aaron; Chen, Ke; Tebben, Andrew; Rampulla, Richard; Wu, Dauh-Rurng; Zhang, Yingru; Mathur, Arvind; White, Ronald; Rose, Anne; Wang, Haiqing; Yang, Zheng; Ranasinghe, Asoka; D'Arienzo, Celia; Guarino, Victor; Xiao, Lan; Su, Ching; Everlof, Gerry; Arora, Vinod; Shen, Ding Ren; Cvijic, Mary Ellen; Menard, Krista; Wen, Mei-Li; Meredith, Jere; Trainor, George; Lombardo, Louis J; Olson, Richard; Baran, Phil S; Hunt, John T; Vite, Gregory D; Fischer, Bruce S; Westhouse, Richard A; Lee, Francis Y

Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms

发现一种高选择性JAK2抑制剂BMS-911543,用于治疗骨髓增生性肿瘤

Wan, Honghe; Schroeder, Gretchen M; Hart, Amy C; Inghrim, Jennifer; Grebinski, James; Tokarski, John S; Lorenzi, Matthew V; You, Dan; Mcdevitt, Theresa; Penhallow, Becky; Vuppugalla, Ragini; Zhang, Yueping; Gu, Xiaomei; Iyer, Ramaswamy; Lombardo, Louis J; Trainor, George L; Ruepp, Stefan; Lippy, Jonathan; Blat, Yuval; Sack, John S; Khan, Javed A; Stefanski, Kevin; Sleczka, Bogdan; Mathur, Arvind; Sun, Jung-Hui; Wong, Michael K; Wu, Dauh-Rurng; Li, Peng; Gupta, Anuradha; Arunachalam, P N; Pragalathan, Bala; Narayanan, Sankara; K C, Nanjundaswamy; Kuppusamy, Prakasam; Purandare, Ashok V