Discovery of RG7388, a potent and selective p53-MDM2 inhibitor in clinical development
发现 RG7388,一种强效且选择性的 p53-MDM2 抑制剂,目前正处于临床开发阶段
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm400487c
Qingjie Ding, Zhuming Zhang, Jin-Jun Liu, Nan Jiang, Jing Zhang, Tina M Ross, Xin-Jie Chu, David Bartkovitz, Frank Podlaski, Cheryl Janson, Christian Tovar, Zoran M Filipovic, Brian Higgins, Kelli Glenn, Kathryn Packman, Lyubomir T Vassilev, Bradford Graves