日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro activity of a G-quadruplex-stabilizing small molecule that synergizes with Navitoclax to induce cytotoxicity in acute myeloid leukemia cells

G-四链体稳定小分子与 Navitoclax 协同作用,在急性髓系白血病细胞中诱导细胞毒性的体外活性

Justin J Montoya, Megan A Turnidge, Daniel H Wai, Apurvi R Patel, David W Lee, Vijay Gokhale, Laurence H Hurley, Robert J Arceci, Cynthia Wetmore, David O Azorsa

Disulfiram overcomes bortezomib and cytarabine resistance in Down-syndrome-associated acute myeloid leukemia cells

双硫仑可克服唐氏综合症相关急性髓系白血病细胞对硼替佐米和阿糖胞苷的耐药性

Ranjan Bista, David W Lee, Oliver B Pepper, David O Azorsa, Robert J Arceci, Eiman Aleem

Aurora B kinase is a potent and selective target in MYCN-driven neuroblastoma

Aurora B 激酶是 MYCN 驱动的神经母细胞瘤的一个有效且有选择性的靶点

Dominik Bogen, Jun S Wei, David O Azorsa, Pinar Ormanoglu, Eugen Buehler, Rajarshi Guha, Jonathan M Keller, Lesley A Mathews Griner, Marc Ferrer, Young K Song, Hongling Liao, Arnulfo Mendoza, Berkley E Gryder, Sivasish Sindri, Jianbin He, Xinyu Wen, Shile Zhang, John F Shern, Marielle E Yohe, Sabine

RNAi screening of the kinome with cytarabine in leukemias

利用阿糖胞苷对白血病中的激酶组进行 RNAi 筛选

Raoul Tibes, James M Bogenberger, Leena Chaudhuri, R Tanner Hagelstrom, Donald Chow, Megan E Buechel, Irma M Gonzales, Tim Demuth, James Slack, Ruben A Mesa, Esteban Braggio, Hongwei H Yin, Shilpi Arora, David O Azorsa

Foxo3a drives proliferation in anaplastic thyroid carcinoma through transcriptional regulation of cyclin A1: a paradigm shift that impacts current therapeutic strategies

Foxo3a 通过转录调控细胞周期蛋白 A1 来驱动未分化甲状腺癌的增殖:影响当前治疗策略的范式转变

Laura A Marlow, Christina A von Roemeling, Simon J Cooper, Yilin Zhang, Stephen D Rohl, Shilpi Arora, Irma M Gonzales, David O Azorsa, Honey V Reddi, Han W Tun, Heike R Döppler, Peter Storz, Robert C Smallridge, John A Copland

Synthetic lethal RNAi screening identifies sensitizing targets for gemcitabine therapy in pancreatic cancer

合成致死 RNAi 筛选确定胰腺癌吉西他滨治疗的敏感靶点

David O Azorsa, Irma M Gonzales, Gargi D Basu, Ashish Choudhary, Shilpi Arora, Kristen M Bisanz, Jeffrey A Kiefer, Meredith C Henderson, Jeffrey M Trent, Daniel D Von Hoff, Spyro Mousses