日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mutations in the Plasmodium falciparum Cyclic Amine Resistance Locus (PfCARL) Confer Multidrug Resistance

恶性疟原虫环胺抗性基因座 (PfCARL) 突变导致多重耐药性

Gregory LaMonte, Michelle Yi-Xiu Lim, Melanie Wree, Christin Reimer, Marie Nachon, Victoria Corey, Peter Gedeck, David Plouffe, Alan Du, Nelissa Figueroa, Bryan Yeung, Pablo Bifani, Elizabeth A Winzeler

High-Throughput Luciferase-Based Assay for the Discovery of Therapeutics That Prevent Malaria

基于高通量荧光素酶的检测方法用于发现预防疟疾的治疗方法

Justine Swann, Victoria Corey, Christina A Scherer, Nobutaka Kato, Eamon Comer, Micah Maetani, Yevgeniya Antonova-Koch, Christin Reimer, Kerstin Gagaring, Maureen Ibanez, David Plouffe, Anne-Marie Zeeman, Clemens H M Kocken, Case W McNamara, Stuart L Schreiber, Brice Campo, Elizabeth A Winzeler, Ste

KAF156 is an antimalarial clinical candidate with potential for use in prophylaxis, treatment, and prevention of disease transmission

KAF156 是一种抗疟临床候选药物,具有用于预防、治疗和防止疾病传播的潜力。

Kelli L Kuhen, Arnab K Chatterjee, Matthias Rottmann, Kerstin Gagaring, Rachel Borboa, Jennifer Buenviaje, Zhong Chen, Carolyn Francek, Tao Wu, Advait Nagle, S Whitney Barnes, David Plouffe, Marcus C S Lee, David A Fidock, Wouter Graumans, Marga van de Vegte-Bolmer, Geert J van Gemert, Grennady Wirj

Imidazolopiperazines: lead optimization of the second-generation antimalarial agents

咪唑并哌嗪类:第二代抗疟药物的先导优化

Advait Nagle, Tao Wu, Kelli Kuhen, Kerstin Gagaring, Rachel Borboa, Caroline Francek, Zhong Chen, David Plouffe, Xuena Lin, Christopher Caldwell, Jared Ek, Suzanne Skolnik, Fenghua Liu, Jianling Wang, Jonathan Chang, Chun Li, Bo Liu, Thomas Hollenbeck, Tove Tuntland, John Isbell, Tiffany Chuan, Phil

Imidazolopiperazines: hit to lead optimization of new antimalarial agents

咪唑并哌嗪:引领新型抗疟药物优化的热门话题

Tao Wu, Advait Nagle, Kelli Kuhen, Kerstin Gagaring, Rachel Borboa, Caroline Francek, Zhong Chen, David Plouffe, Anne Goh, Suresh B Lakshminarayana, Jeanette Wu, Hui Qing Ang, Peiting Zeng, Min Low Kang, William Tan, Maria Tan, Nicole Ye, Xuena Lin, Christopher Caldwell, Jared Ek, Suzanne Skolnik, F

A systematic approach to understand the mechanism of action of the bisthiazolium compound T4 on the human malaria parasite, Plasmodium falciparum

系统地了解双噻唑化合物 T4 对人类疟原虫恶性疟原虫的作用机制

Karine G Le Roch, Jeffrey R Johnson, Hugues Ahiboh, Duk-Won D Chung, Jacques Prudhomme, David Plouffe, Kerstin Henson, Yingyao Zhou, William Witola, John R Yates, Choukri Ben Mamoun, Elizabeth A Winzeler, Henri Vial

Evidence-based annotation of the malaria parasite's genome using comparative expression profiling

使用比较表达谱对疟原虫基因组进行循证注释

Yingyao Zhou, Vandana Ramachandran, Kota Arun Kumar, Scott Westenberger, Phillippe Refour, Bin Zhou, Fengwu Li, Jason A Young, Kaisheng Chen, David Plouffe, Kerstin Henson, Victor Nussenzweig, Jane Carlton, Joseph M Vinetz, Manoj T Duraisingh, Elizabeth A Winzeler