日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Activation of CAMK2 by pseudokinase PEAK1 represents a targetable pathway in triple negative breast cancer

假激酶 PEAK1 激活 CAMK2 是三阴性乳腺癌中可靶向的通路

Xue Yang, Xiuquan Ma, Tianyue Zhao, David R Croucher, Elizabeth V Nguyen, Kimberley C Clark, Changyuan Hu, Sharissa L Latham, Charles Bayly-Jones, Bao V Nguyen, Srikanth Budnar, Sung-Young Shin, Lan K Nguyen, Thomas R Cotton, Anderly C Chüeh, Terry C C Lim Kam Sian, Margaret M Stratton, Andrew M Ell

A first-in-class pan-lysyl oxidase inhibitor impairs stromal remodeling and enhances gemcitabine response and survival in pancreatic cancer

一种首创的泛赖氨酰氧化酶抑制剂可抑制基质重塑,并增强吉西他滨对胰腺癌的疗效和生存率。

Jessica L Chitty,Michelle Yam #,Lara Perryman #,Amelia L Parker,Joanna N Skhinas,Yordanos F I Setargew,Ellie T Y Mok,Emmi Tran,Rhiannon D Grant,Sharissa L Latham ,Brooke A Pereira ,Shona C Ritchie,Kendelle J Murphy ,Michael Trpceski ,Alison D Findlay,Pauline Melenec,Elysse C Filipe,Audrey Nadalini,Sipiththa Velayuthar,Gretel Major,Kaitlin Wyllie,Michael Papanicolaou,Shivanjali Ratnaseelan,Phoebe A Phillips,George Sharbeen,Janet Youkhana,Alice Russo,Antonia Blackwell,Jordan F Hastings,Morghan C Lucas,Cecilia R Chambers,Daniel A Reed,Janett Stoehr,Claire Vennin,Ruth Pidsley ,Anaiis Zaratzian,Andrew M Da Silva,Michael Tayao,Brett Charlton,David Herrmann,Max Nobis ,Susan J Clark ,Andrew V Biankin ,Amber L Johns,David R Croucher ,Adnan Nagrial,Anthony J Gill   ,Sean M Grimmond  ; Australian Pancreatic Cancer Genome Initiative (APGI); Australian Pancreatic Cancer Matrix Atlas (APMA); Marina Pajic ,Paul Timpson,Wolfgang Jarolimek,Thomas R Cox

Mepolizumab decreases tissue eosinophils while increasing type-2 cytokines in eosinophilic chronic rhinosinusitis

美泊利单抗可减少嗜酸性慢性鼻窦炎中的组织嗜酸性粒细胞,同时增加 2 型细胞因子

Sophie Walter, Jacqueline Ho, Raquel Alvarado, Greg Smith, David R Croucher, Sharron Liang, Jessica W Grayson, João Mangussi-Gomes, Simone L Van Es, Peter Earls, Janet Rimmer, Raewyn Campbell, Larry Kalish, Raymond Sacks, Richard J Harvey

Prostate cancer cell proliferation is influenced by LDL-cholesterol availability and cholesteryl ester turnover

前列腺癌细胞增殖受低密度脂蛋白胆固醇利用率和胆固醇酯周转率的影响

Nikki L Raftopulos #, Tinashe C Washaya #, Andreas Niederprüm, Antonia Egert, Mariam F Hakeem-Sanni, Bianca Varney, Atqiya Aishah, Mariya L Georgieva, Ellinor Olsson, Diandra Z Dos Santos, Zeyad D Nassar, Blake J Cochran, Shilpa R Nagarajan, Meghna S Kakani, Jordan F Hastings, David R Croucher, Kerr

A non-genetic, cell cycle-dependent mechanism of platinum resistance in lung adenocarcinoma

肺腺癌铂类耐药的非遗传、细胞周期依赖性机制

Alvaro Gonzalez Rajal, Kamila A Marzec, Rachael A McCloy, Max Nobis, Venessa Chin, Jordan F Hastings, Kaitao Lai, Marina Kennerson, William E Hughes, Vijesh Vaghjiani, Paul Timpson, Jason E Cain, D Neil Watkins, David R Croucher #, Andrew Burgess #

Bisphosphonate drugs have actions in the lung and inhibit the mevalonate pathway in alveolar macrophages

双膦酸盐类药物在肺部发挥作用,抑制肺泡巨噬细胞中的甲羟戊酸途径。

Marcia A Munoz ,Emma K Fletcher ,Oliver P Skinner ,Julie Jurczyluk ,Esther Kristianto ,Mark P Hodson ,Shuting Sun ,Frank H Ebetino ,David R Croucher ,Philip M Hansbro ,Jacqueline R Center ,Michael J Rogers

Analysis of pulsed cisplatin signalling dynamics identifies effectors of resistance in lung adenocarcinoma

脉冲顺铂信号动力学分析可识别肺腺癌的耐药效应物

Jordan F Hastings #, Alvaro Gonzalez Rajal #, Sharissa L Latham, Jeremy Zr Han, Rachael A McCloy, Yolande Ei O'Donnell, Monica Phimmachanh, Alexander D Murphy, Adnan Nagrial, Dariush Daneshvar, Venessa Chin, D Neil Watkins, Andrew Burgess, David R Croucher

Structure-based mechanism of preferential complex formation by apoptosis signal-regulating kinases

凋亡信号调节激酶优先形成复合物的结构机制

Sarah J Trevelyan, Jodi L Brewster, Abigail E Burgess, Jennifer M Crowther, Antonia L Cadell, Benjamin L Parker, David R Croucher, Renwick C J Dobson, James M Murphy, Peter D Mace

A cryptic tubulin-binding domain links MEKK1 to curved tubulin protomers

隐秘的微管蛋白结合域将 MEKK1 与弯曲的微管蛋白原体连接起来

Pavel Filipčík, Sharissa L Latham, Antonia L Cadell, Catherine L Day, David R Croucher, Peter D Mace

PP1 initiates the dephosphorylation of MASTL, triggering mitotic exit and bistability in human cells

PP1 启动 MASTL 的去磷酸化,引发人类细胞中有丝分裂退出和双稳态

Samuel Rogers, Dirk Fey, Rachael A McCloy, Benjamin L Parker, Nicholas J Mitchell, Richard J Payne, Roger J Daly, David E James, C Elizabeth Caldon, D Neil Watkins, David R Croucher, Andrew Burgess