日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Collateral lethality between HDAC1 and HDAC2 exploits cancer-specific NuRD complex vulnerabilities

HDAC1 和 HDAC2 之间的附带致死性利用了癌症特异性 NuRD 复合物的脆弱性

Yuxiang Zhang, David Remillard, Ugoma Onubogu, Barbara Karakyriakou, Joshua N Asiaban, Anissa R Ramos, Kirsten Bowland, Timothy R Bishop, Paige A Barta, Stephanie Nance, Adam D Durbin, Christopher J Ott, Michalina Janiszewska, Benjamin F Cravatt, Michael A Erb

A novel β-catenin/BCL9 complex inhibitor blocks oncogenic Wnt signaling and disrupts cholesterol homeostasis in colorectal cancer

新型 β-catenin/BCL9 复合物抑制剂可阻断致癌 Wnt 信号并破坏结直肠癌中的胆固醇稳态

Helen Tanton, Tomasz Sewastianik, Hyuk-Soo Seo, David Remillard, Roodolph St Pierre, Pratyusha Bala, Daulet Aitymbayev, Peter Dennis, Keith Adler, Ezekiel Geffken, Zoe Yeoh, Nicholas Vangos, Filip Garbicz, David Scott, Nilay Sethi, James Bradner, Sirano Dhe-Paganon, Ruben D Carrasco

An Activity-Guided Map of Electrophile-Cysteine Interactions in Primary Human T Cells

人类原代 T 细胞中亲电试剂-半胱氨酸相互作用的活性引导图谱

Ekaterina V Vinogradova, Xiaoyu Zhang, David Remillard, Daniel C Lazar, Radu M Suciu, Yujia Wang, Giulia Bianco, Yu Yamashita, Vincent M Crowley, Michael A Schafroth, Minoru Yokoyama, David B Konrad, Kenneth M Lum, Gabriel M Simon, Esther K Kemper, Michael R Lazear, Sifei Yin, Megan M Blewett, Melis

Targeted degradation of BRD9 reverses oncogenic gene expression in synovial sarcoma

靶向降解BRD9可逆转滑膜肉瘤中的致癌基因表达

Gerard L Brien ,David Remillard ,Junwei Shi ,Matthew L Hemming ,Jonathon Chabon ,Kieran Wynne ,Eugène T Dillon ,Gerard Cagney ,Guido Van Mierlo ,Marijke P Baltissen ,Michiel Vermeulen ,Jun Qi ,Stefan Fröhling ,Nathanael S Gray ,James E Bradner ,Christopher R Vakoc ,Scott A Armstrong

Degradation of the BAF Complex Factor BRD9 by Heterobifunctional Ligands

异双功能配体降解 BAF 复合物因子 BRD9

David Remillard, Dennis L Buckley, Joshiawa Paulk, Gerard L Brien, Matthew Sonnett, Hyuk-Soo Seo, Shiva Dastjerdi, Martin Wühr, Sirano Dhe-Paganon, Scott A Armstrong, James E Bradner

Influence of attitudes toward curriculum on dishonest academic behavior

对课程的态度对学术不端行为的影响

Austin, Zubin; Collins, David; Remillard, Alfred; Kelcher, Sheila; Chui, Stephanie