日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fabry disease: a rare disorder calling for personalized medicine

法布里病:一种罕见疾病,亟需个性化医疗

Lerario, Sarah; Monti, Luigi; Ambrosetti, Irene; Luglio, Agnese; Pietra, Andrea; Aiello, Valeria; Montanari, Francesca; Bellasi, Antonio; Zaza, Gianluigi; Galante, Antonio; Salera, Davide; Capelli, Irene; La Manna, Gaetano; Provenzano, Michele

Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the β-Catenin Armadillo Repeats Domain as an Anticancer Agent

新型N-(杂环苯基)苯磺酰胺与T细胞因子4在β-catenin Armadillo重复结构域共享一个未报道的结合位点,可作为抗癌剂

Marianna Nalli ,Laura Di Magno ,Yichao Wen ,Xin Liu ,Michele D'Ambrosio ,Michela Puxeddu ,Anastasia Parisi ,Jessica Sebastiani ,Andrea Sorato ,Antonio Coluccia ,Silvia Ripa ,Fiorella Di Pastena ,Davide Capelli ,Roberta Montanari ,Domiziana Masci ,Andrea Urbani ,Chiara Naro ,Claudio Sette ,Viviana Orlando ,Sara D'Angelo ,Stefano Biagioni ,Chiara Bigogno ,Giulio Dondio ,Arianna Pastore ,Mariano Stornaiuolo ,Gianluca Canettieri ,Te Liu ,Romano Silvestri ,Giuseppe La Regina

Biological Screening and Crystallographic Studies of Hydroxy γ-Lactone Derivatives to Investigate PPARγ Phosphorylation Inhibition

羟基 γ-内酯衍生物的生物筛选和晶体学研究以探究 PPARγ 磷酸化抑制作用

Davide Capelli, Giulia Cazzaniga, Matteo Mori, Antonio Laghezza, Fulvio Loiodice, Martina Quaglia, Elisa Negro, Fiorella Meneghetti, Stefania Villa, Roberta Montanari

Cytosolic localization and in vitro assembly of human de novo thymidylate synthesis complex

人类胸苷酸从头合成复合物的细胞质定位和体外组装

Sharon Spizzichino, Dalila Boi, Giovanna Boumis, Roberta Lucchi, Francesca Romana Liberati, Davide Capelli, Roberta Montanari, Giorgio Pochetti, Roberta Piacentini, Giacomo Parisi, Alessio Paone, Serena Rinaldo, Roberto Contestabile, Angela Tramonti, Alessandro Paiardini, Giorgio Giardina, Francesca

PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc

PHA-680626 是 Aurora-A 与 N-Myc 相互作用的有效抑制剂

Dalila Boi, Fani Souvalidou, Davide Capelli, Federica Polverino, Grazia Marini, Roberta Montanari, Giorgio Pochetti, Angela Tramonti, Roberto Contestabile, Daniela Trisciuoglio, Patrizia Carpinelli, Camilla Ascanelli, Catherine Lindon, Alessandro De Leo, Michele Saviano, Roberto Di Santo, Roberta Co

Discovery of Novel Chemical Series of OXA-48 β-Lactamase Inhibitors by High-Throughput Screening

通过高通量筛选发现一系列新型 OXA-48 β-内酰胺酶抑制剂

Barbara Garofalo, Federica Prati, Rosa Buonfiglio, Isabella Coletta, Noemi D'Atanasio, Angela Molteni, Daniele Carettoni, Valeria Wanke, Giorgio Pochetti, Roberta Montanari, Davide Capelli, Claudio Milanese, Francesco Paolo Di Giorgio, Rosella Ombrato

A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities

一种具有独特过氧化物酶体增殖激活受体γ结合特性和生物活性的新型N取代缬氨酸衍生物

Franck Peiretti, Roberta Montanari, Davide Capelli, Bernadette Bonardo, Cécilia Colson, Ez-Zoubir Amri, Marina Grimaldi, Patrick Balaguer, Keiichi Ito, Robert G Roeder, Giorgio Pochetti, Jean Michel Brunel

Swarm-CG: Automatic Parametrization of Bonded Terms in MARTINI-Based Coarse-Grained Models of Simple to Complex Molecules via Fuzzy Self-Tuning Particle Swarm Optimization

Swarm-CG:基于模糊自整定粒子群优化算法的MARTINI粗粒化模型中简单到复杂分子键合项的自动参数化

Empereur-Mot, Charly; Pesce, Luca; Doni, Giovanni; Bochicchio, Davide; Capelli, Riccardo; Perego, Claudio; Pavan, Giovanni M

Surface Plasmon Resonance as a Tool for Ligand Binding Investigation of Engineered GPR17 Receptor, a G Protein Coupled Receptor Involved in Myelination

表面等离子体共振作为配体结合研究的工具,研究工程化 GPR17 受体(一种参与髓鞘形成的 G 蛋白偶联受体)

Davide Capelli, Chiara Parravicini, Giorgio Pochetti, Roberta Montanari, Caterina Temporini, Marco Rabuffetti, Maria Letizia Trincavelli, Simona Daniele, Marta Fumagalli, Simona Saporiti, Elisabetta Bonfanti, Maria P Abbracchio, Ivano Eberini, Stefania Ceruti, Enrica Calleri, Stefano Capaldi

Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode

新型配体结合模式揭示 PPAR 部分或完全激活的结构基础

Davide Capelli, Carmen Cerchia, Roberta Montanari, Fulvio Loiodice, Paolo Tortorella, Antonio Laghezza, Laura Cervoni, Giorgio Pochetti, Antonio Lavecchia