日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of RXFP2 genetic association in resistant hypertensive men and RXFP2 antagonists for the treatment of resistant hypertension

发现RXFP2基因与难治性高血压男性患者相关,以及RXFP2拮抗剂在治疗难治性高血压中的应用

Shan-Shan Zhang #,Lance Larrabee #,Andrew H Chang,Sapna Desai,Lisa Sloan,Xin Wang,Yixuan Wu,Nazia Parvez,Karen Amaratunga,Allison C Hartman,Abby Whitnall,Joseph Mason,Nicholas P Barton,Audrey Y Chu,Jonathan M Davitte,Adam J Csakai,Caitlin Vestal Tibbetts,Audrey E Tolbert,Heather O'Keefe,Jessie Polanco,Joseph Foley,Casey Kmett,Jonathan Kehler,Gabriela Kozejova,Feng Wang,Andrew P Mayer,Patrick Koenig,Davide Foletti,Steven J Pitts,Christine G Schnackenberg

Targeting CLDN18.2 by CD3 Bispecific and ADC Modalities for the Treatments of Gastric and Pancreatic Cancer

通过 CD3 双特异性和 ADC 方式靶向 CLDN18.2 治疗胃癌和胰腺癌

Guoyun Zhu, Davide Foletti, Xiaohui Liu, Sheng Ding, Jody Melton Witt, Adela Hasa-Moreno, Mathias Rickert, Charles Holz, Laura Aschenbrenner, Amy H Yang, Eugenia Kraynov, Winston Evering, Leslie Obert, Chenyu Lee, Tao Sai, Tina Mistry, Kevin C Lindquist, Thomas Van Blarcom, Pavel Strop, Javier Chapa

Germline-encoded neutralization of a Staphylococcus aureus virulence factor by the human antibody repertoire

人类抗体库对金黄色葡萄球菌毒力因子的种系编码中和

Yik Andy Yeung, Davide Foletti, Xiaodi Deng, Yasmina Abdiche, Pavel Strop, Jacob Glanville, Steven Pitts, Kevin Lindquist, Purnima D Sundar, Marina Sirota, Adela Hasa-Moreno, Amber Pham, Jody Melton Witt, Irene Ni, Jaume Pons, David Shelton, Arvind Rajpal, Javier Chaparro-Riggers

Production of soluble and active microbial transglutaminase in Escherichia coli for site-specific antibody drug conjugation

大肠杆菌中生产可溶活性微生物转谷氨酰胺酶用于位点特异性抗体药物结合

Mathias Rickert, Pavel Strop, Victor Lui, Jody Melton-Witt, Santiago Esteban Farias, Davide Foletti, David Shelton, Jaume Pons, Arvind Rajpal

Engineering Highly Potent and Selective Microproteins against Nav1.7 Sodium Channel for Treatment of Pain

针对 Nav1.7 钠通道设计高效选择性微蛋白用于治疗疼痛

Anatoly Shcherbatko, Andrea Rossi, Davide Foletti, Guoyun Zhu, Oren Bogin, Meritxell Galindo Casas, Mathias Rickert, Adela Hasa-Moreno, Victor Bartsevich, Andreas Crameri, Alexander R Steiner, Robert Henningsen, Avinash Gill, Jaume Pons, David L Shelton, Arvind Rajpal, Pavel Strop

Site-Dependent Degradation of a Non-Cleavable Auristatin-Based Linker-Payload in Rodent Plasma and Its Effect on ADC Efficacy

啮齿动物血浆中不可裂解的基于 Auristatin 的连接子-有效载荷的位点依赖性降解及其对 ADC 疗效的影响

Magdalena Dorywalska, Pavel Strop, Jody A Melton-Witt, Adela Hasa-Moreno, Santiago E Farias, Meritxell Galindo Casas, Kathy Delaria, Victor Lui, Kris Poulsen, Janette Sutton, Gary Bolton, Dahui Zhou, Ludivine Moine, Russell Dushin, Thomas-Toan Tran, Shu-Hui Liu, Mathias Rickert, Davide Foletti, Davi

Generation of a high-fidelity antibody against nerve growth factor using library scanning mutagenesis and validation with structures of the initial and optimized Fab-antigen complexes

使用文库扫描诱变生成针对神经生长因子的高保真抗体并使用初始和优化的 Fab-抗原复合物的结构进行验证

Sherry L La Porte, Charles Eigenbrot, Mark Ultsch, Wei-Hsien Ho, Davide Foletti, Alison Forgie, Kevin C Lindquist, David L Shelton, Jaume Pons

High-throughput epitope binning assays on label-free array-based biosensors can yield exquisite epitope discrimination that facilitates the selection of monoclonal antibodies with functional activity

在无标记阵列生物传感器上进行高通量表位分类分析可以产生精确的表位鉴别,从而有助于选择具有功能活性的单克隆抗体

Yasmina Noubia Abdiche, Adam Miles, Josh Eckman, Davide Foletti, Thomas J Van Blarcom, Yik Andy Yeung, Jaume Pons, Arvind Rajpal