日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into the unexpected agonism of tetracyclic antidepressants at serotonin receptors 5-HT1eR and 5-HT1FR

四环抗抑郁药对血清素受体 5-HT1eR 和 5-HT1FR 的意外激动作用的结构洞察

Gregory Zilberg, Alexandra K Parpounas, Audrey L Warren, Bianca Fiorillo, Davide Provasi, Marta Filizola, Daniel Wacker

Gαs slow conformational transition upon GTP binding and a novel Gαs regulator

Gαs 在 GTP 结合时的缓慢构象转变和一种新型 Gαs 调节剂

Donghoon Ahn, Davide Provasi, Nguyen Minh Duc, Jun Xu, Leslie Salas-Estrada, Aleksandar Spasic, Min Woo Yun, Juyeong Kang, Dongmin Gim, Jaecheol Lee, Yang Du, Marta Filizola, Ka Young Chung

A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects

一种具有低效 Mu 阿片受体激动作用的新型 Mitragynine 类似物表现出抗伤害作用,且不良反应减弱

Soumen Chakraborty, Jeffrey F DiBerto, Abdelfattah Faouzi, Sarah M Bernhard, Anna M Gutridge, Steven Ramsey, Yuchen Zhou, Davide Provasi, Nitin Nuthikattu, Rahul Jilakara, Melissa N F Nelson, Wesley B Asher, Shainnel O Eans, Lisa L Wilson, Satyanarayana M Chintala, Marta Filizola, Richard M van Rijn

Differences in interactions between transmembrane domains tune the activation of metabotropic glutamate receptors

跨膜结构域之间相互作用的差异调节代谢型谷氨酸受体的激活

Jordana K Thibado, Jean-Yves Tano, Joon Lee, Leslie Salas-Estrada, Davide Provasi, Alexa Strauss, Joao Marcelo Lamim Ribeiro, Guoqing Xiang, Johannes Broichhagen, Marta Filizola, Martin J Lohse, Joshua Levitz

Development of novel biosensors to study receptor-mediated activation of the G-protein α subunits Gs and Golf

开发新型生物传感器来研究受体介导的 G 蛋白 α 亚基 Gs 和 Golf 的激活

Hideaki Yano, Davide Provasi, Ning Sheng Cai, Marta Filizola, Sergi Ferré, Jonathan A Javitch