日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Olaparib increases the therapeutic index of hemithoracic irradiation compared with hemithoracic irradiation alone in a mouse lung cancer model

在小鼠肺癌模型中,与单独进行半胸照射相比,奥拉帕尼可提高半胸照射的治疗指数。

Jiang, Yanyan; Martin, Jennifer; Alkadhimi, Maryam; Shigemori, Kay; Kinchesh, Paul; Gilchrist, Stuart; Kersemans, Veerle; Smart, Sean; Thompson, James M; Hill, Mark A; O'Connor, Mark J; Davies, Barry R; Ryan, Anderson J

Design and optimisation of dendrimer-conjugated Bcl-2/x(L) inhibitor, AZD0466, with improved therapeutic index for cancer therapy

设计和优化树状聚合物偶联的Bcl-2/x(L)抑制剂AZD0466,以提高其在癌症治疗中的治疗指数

Patterson, Claire M; Balachander, Srividya B; Grant, Iain; Pop-Damkov, Petar; Kelly, Brian; McCoull, William; Parker, Jeremy; Giannis, Michael; Hill, Kathryn J; Gibbons, Francis D; Hennessy, Edward J; Kemmitt, Paul; Harmer, Alexander R; Gales, Sonya; Purbrick, Stuart; Redmond, Sean; Skinner, Matthew; Graham, Lorraine; Secrist, J Paul; Schuller, Alwin G; Wen, Shenghua; Adam, Ammar; Reimer, Corinne; Cidado, Justin; Wild, Martin; Gangl, Eric; Fawell, Stephen E; Saeh, Jamal; Davies, Barry R; Owen, David J; Ashford, Marianne B

Genetic Alterations in the PI3K/AKT Pathway and Baseline AKT Activity Define AKT Inhibitor Sensitivity in Breast Cancer Patient-derived Xenografts

PI3K/AKT通路中的基因改变和基线AKT活性决定了乳腺癌患者来源异种移植瘤对AKT抑制剂的敏感性

Gris-Oliver, Albert; Palafox, Marta; Monserrat, Laia; Brasó-Maristany, Fara; Òdena, Andreu; Sánchez-Guixé, Mònica; Ibrahim, Yasir H; Villacampa, Guillermo; Grueso, Judit; Parés, Mireia; Guzmán, Marta; Rodríguez, Olga; Bruna, Alejandra; Hirst, Caroline S; Barnicle, Alan; de Bruin, Elza C; Reddy, Avinash; Schiavon, Gaia; Arribas, Joaquín; Mills, Gordon B; Caldas, Carlos; Dienstmann, Rodrigo; Prat, Aleix; Nuciforo, Paolo; Razavi, Pedram; Scaltriti, Maurizio; Turner, Nicholas C; Saura, Cristina; Davies, Barry R; Oliveira, Mafalda; Serra, Violeta

Optimizing the design of population-based patient-derived tumor xenograft studies to better predict clinical response

优化基于人群的患者来源肿瘤异种移植研究设计,以更好地预测临床反应

Floc'h, Nicolas; Guerriero, Maria Luisa; Ramos-Montoya, Antonio; Davies, Barry R; Cairns, Jonathan; Karp, Natasha A

Akt inhibition improves long-term tumour control following radiotherapy by altering the microenvironment

Akt抑制剂通过改变肿瘤微环境,改善放疗后肿瘤的长期控制。

Searle, Emma J; Telfer, Brian A; Mukherjee, Debayan; Forster, Duncan M; Davies, Barry R; Williams, Kaye J; Stratford, Ian J; Illidge, Tim M

Efficacy of targeted AKT inhibition in genetically engineered mouse models of PTEN-deficient prostate cancer

靶向AKT抑制在PTEN缺陷型前列腺癌基因工程小鼠模型中的疗效

De Velasco, Marco A; Kura, Yurie; Yoshikawa, Kazuhiro; Nishio, Kazuto; Davies, Barry R; Uemura, Hirotsugu

Autophagy limits the cytotoxic effects of the AKT inhibitor AZ7328 in human bladder cancer cells.

自噬限制了 AKT 抑制剂 AZ7328 对人类膀胱癌细胞的细胞毒性作用

Dickstein Rian J, Nitti Giovanni, Dinney Colin P, Davies Barry R, Kamat Ashish M, McConkey David J