日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents

奥司他韦氮丙啶类药物是强效的流感神经氨酸酶抑制剂和显像剂。

Vriends, Merijn B L; Moran, Elisha; Calvelo, Martín; Hansen, Thomas; Pickles, Isabelle B; Xin, Xincheng; Biezeno, Marieke; Armstrong, Zachary W B; Ferraz, Maria J; Li, Lei; Lilley, Alice; Harvey, Ruth; Filippov, Dmitri V; Liao, Qinghua; Schröder, Sybrin P; van der Marel, Gijsbert A; Artola, Marta; Aerts, Johannes M F G; Blaza, James N; Codée, Jeroen D C; Rovira, Carme; Overkleeft, Herman S; Davies, Gideon J

Signal-strapping as a protein-sequence search method for the discovery of metalloproteins

信号绑扎法作为一种蛋白质序列搜索方法,用于发现金属蛋白

Franco Cairo, João Paulo L; Corrêa, Thamy L R; Offen, Wendy A; Nairn, Alison K; Walton, Julia; Sweeney, Sean T; Davies, Gideon J; Walton, Paul H

Bespoke Activity-Based Probes Reveal that the Pseudomonas aeruginosa Endoglycosidase, PslG, Is an Endo-β-glucanase

定制的活性探针揭示铜绿假单胞菌内切糖苷酶 PslG 是一种内切β-葡聚糖酶

Ruijgrok, Gijs; Offen, Wendy A; Pickles, Isabelle B; Raju, Deepa; Patsos, Thanasis; de Boer, Casper; Ofman, Tim; Rompa, Joep; van Oord, Daan; Dodson, Eleanor J; Beekers, Alexander; Voskuilen, Thijs; Ferrari, Michela; Wu, Liang; Janssen, Antonius P A; Codée, Jeroen D C; Howell, P Lynne; Davies, Gideon J; Overkleeft, Herman S

Design, modular synthesis and screening of 58 shape-diverse 3-D fragments

设计、模块化合成和筛选58种形状各异的三维片段

Downes, Thomas D; Jones, S Paul; Firth, James D; Darby, John F; Gilio, Amelia K; Klein, Hanna F; Wang, Xinyu; Blakemore, David C; De Fusco, Claudia; Roughley, Stephen D; Vidler, Lewis R; Whatton, Maria Ann; Woolford, Alison J-A; Wrigley, Gail L; Hubbard, Roderick E; Wu, Liang; Davies, Gideon J; O'Brien, Peter

Structure, kinetics, and mechanism of Pseudomonas putida sulfoquinovose dehydrogenase, the first enzyme in the sulfoglycolytic Entner-Doudoroff pathway

假单胞菌磺基喹诺糖脱氢酶的结构、动力学和机制,该酶是磺基糖酵解Entner-Doudoroff途径中的第一个酶。

Burchill, Laura; Sharma, Mahima; Soler, Niccolay Madiedo; Goddard-Borger, Ethan D; Davies, Gideon J; Williams, Spencer J

Activity-based probes for dynamic characterisation of polysaccharide-degrading enzymes

用于动态表征多糖降解酶的活性探针

Pickles, Isabelle B; Corrêa, Thamy L R; Overkleeft, Herman S; Davies, Gideon J

Sulfoglycolysis sustains Eubacterium rectale in low-fiber diets

硫糖分解作用维持着真杆菌在低纤维饮食中的生存

Sharma, Mahima; Pudlo, Nicholas; Järvå, Michael A; Kaur, Arashdeep; John, Alan; Burchill, Laura; Lingford, James P; Epa, Ruwan; Abayakoon, Palika; Scott, Nichollas E; Turkenburg, Johan P; Davies, Gideon J; Martens, Eric C; Goddard-Borger, Ethan D; Williams, Spencer J

Expansion of the diversity of dispersin scaffolds

分散蛋白支架多样性的扩展

Males, Alexandra; Moroz, Olga V; Blagova, Elena; Munch, Astrid; Hansen, Gustav H; Johansen, Annette H; Østergaard, Lars H; Segura, Dorotea R; Eddenden, Alexander; Due, Anne V; Gudmand, Martin; Salomon, Jesper; Sørensen, Sebastian R; Franco Cairo, João Paulo L; Nitz, Mark; Pache, Roland A; Vejborg, Rebecca M; Bhosale, Sandeep; Vocadlo, David J; Davies, Gideon J; Wilson, Keith S

Structures of α-galactosaminidases from the CAZy GH114 family and homologs defining a new GH191 family of glycosidases.

CAZy GH114 家族的 α-半乳糖胺酶及其同源物的结构定义了一个新的 GH191 糖苷酶家族

Roth Christian, Moroz Olga V, Miranda Suzan A D, Jahn Lucas, Blagova Elena V, Lebedev Andrey A, Segura Dorotea R, Stringer Mary A, Friis Esben P, Franco Cairo João P L, Davies Gideon J, Wilson Keith S

From Mechanism-Based Retaining Glycosidase Inhibitors to Activity-Based Glycosidase Profiling

从基于机制的保留型糖苷酶抑制剂到基于活性的糖苷酶谱分析

Artola, Marta; Aerts, Johannes M F G; van der Marel, Gijsbert A; Rovira, Carme; Codée, Jeroen D C; Davies, Gideon J; Overkleeft, Herman S