日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Restoration of the Tumor Suppressor Function of Y220C-Mutant p53 by Rezatapopt, a Small-Molecule Reactivator.

Rezatapopt(一种小分子激活剂)可恢复 Y220C 突变 p53 的肿瘤抑制功能

Puzio-Kuter Anna M, Xu Lizhong, McBrayer Mary Kate, Dominique Romyr, Li Hongju H, Fahr Bruce J, Brown Alyssa M, Wiebesiek Amy E, Russo Brandon M, Mulligan Chris L, Yang Hong, Battaglia Josh, Robell Kimberly A, Thomas Dafydd H, Huang Kuo-Sen, Solovyov Alexander, Greenbaum Benjamin D, Oliner Jonathan D, Davis Thomas W, Dumble Melissa L, Johnson Melissa L, Xiong Shunbin, Yang Peirong, Lozano Guillermina, Fellous Marc M, Vu Binh T, Schram Alison M, Levine Arnold J, Poyurovsky Masha V

Discovery of Rezatapopt (PC14586), a First-in-Class, Small-Molecule Reactivator of p53 Y220C Mutant in Development

发现 Rezatapopt (PC14586),一种首创的小分子 p53 Y220C 突变体激活剂

Vu, Binh T; Dominique, Romyr; Fahr, Bruce J; Li, Hongju H; Fry, David C; Xu, Lizhong; Yang, Hong; Puzio-Kuter, Anna; Good, Andrew; Liu, Binbin; Huang, Kuo-Sen; Tanaka, Naoko; Davis, Thomas W; Dumble, Melissa L

Clinician perspectives on designing and implementing a hereditary cancer transition clinic

临床医生对设计和实施遗传性癌症过渡诊所的看法

Gabriel, Jazmine L; Schlieder, Victoria; Goehringer, Jessica M; Leitzel, Tracey; Sugrue, Emily Ann; Zultevicz, Sarah; Davis, Thomas W; Campbell-Salome, Gemme; Romagnoli, Katrina

Targeted BMI1 inhibition impairs tumor growth in lung adenocarcinomas with low CEBPα expression

靶向抑制BMI1可抑制CEBPα低表达肺腺癌的肿瘤生长

Yong, Kol Jia; Basseres, Daniela S; Welner, Robert S; Zhang, Wen Cai; Yang, Henry; Yan, Benedict; Alberich-Jorda, Meritxell; Zhang, Junyan; de Figueiredo-Pontes, Lorena Lobo; Battelli, Chiara; Hetherington, Christopher J; Ye, Min; Zhang, Hong; Maroni, Giorgia; O'Brien, Karen; Magli, Maria Cristina; Borczuk, Alain C; Varticovski, Lyuba; Kocher, Olivier; Zhang, Pu; Moon, Young-Choon; Sydorenko, Nadiya; Cao, Liangxian; Davis, Thomas W; Thakkar, Bhavin M; Soo, Ross A; Iwama, Atsushi; Lim, Bing; Halmos, Balazs; Neuberg, Donna; Tenen, Daniel G; Levantini, Elena

BMI-1 Targeting Interferes with Patient-Derived Tumor-Initiating Cell Survival and Tumor Growth in Prostate Cancer.

BMI-1靶向治疗干扰前列腺癌患者来源的肿瘤起始细胞的存活和肿瘤生长

Bansal Nitu, Bartucci Monica, Yusuff Shamila, Davis Stephani, Flaherty Kathleen, Huselid Eric, Patrizii Michele, Jones Daniel, Cao Liangxian, Sydorenko Nadiya, Moon Young-Choon, Zhong Hua, Medina Daniel J, Kerrigan John, Stein Mark N, Kim Isaac Y, Davis Thomas W, DiPaola Robert S, Bertino Joseph R, Sabaawy Hatem E