日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of spirodioxolane nsP2 helicase inhibitors with antialphaviral activity

鉴定具有抗甲病毒活性的螺二氧戊环nsP2解旋酶抑制剂

Oh, Hans J; Sears, John D; Ramalingam, Bose Muthu; Saleem, Rahman Shah Zaib; Davis-Gilbert, Zachary W; Hossain, Mohammed Anwar; Moorman, Stella R; Ohja, Durbadal; Martinez, Sabian A; Burdick, Jane E; Couñago, Rafael M; Moorman, Nathaniel J; Heise, Mark T; Todd, Matthew H; Willson, Timothy M

Structural insights into human brachyury DNA recognition and discovery of progressible binders for cancer therapy

对人类短尾蛋白DNA识别的结构性见解以及用于癌症治疗的新型结合剂的发现

Newman, Joseph A; Gavard, Angeline E; Imprachim, Nergis; Aitkenhead, Hazel; Sheppard, Hadley E; Te Poele, Robert; Clarke, Paul A; Hossain, Mohammad Anwar; Temme, Louisa; Oh, Hans J; Wells, Carrow I; Davis-Gilbert, Zachary W; Workman, Paul; Gileadi, Opher; Drewry, David H

Identification of Direct-Acting nsP2 Helicase Inhibitors with Antialphaviral Activity

鉴定具有抗甲病毒活性的直接作用nsP2解旋酶抑制剂

Muthu Ramalingam, Bose; Sears, John D; Talbot, Kacey M; Su, Yuan-Wei Norman; Houliston, Scott; Hossain, Mohammed Anwar; Davis-Gilbert, Zachary W; Zhao, Chunqing; Oh, Hans J; Brown, Peter J; Sanders, Marcia K; Moorman, Stella R; Ojha, Durbadal; Burdick, Jane E; Law, Isabella; Morales, Noah L; Martinez, Sabian A; Loppnau, Peter; Garcia Perez, Julia; Drobish, Adam M; Morrison, Thomas E; Streblow, Zachary J; Streblow, Daniel N; Arrowsmith, Cheryl H; Vargason, Ava; Couñago, Rafael M; Halabelian, Levon; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

NUAK2 is a therapeutically tractable regulator of RNA splicing and tumor progression in neuroendocrine prostate cancer

NUAK2是神经内分泌前列腺癌中RNA剪接和肿瘤进展的一个具有治疗潜力的调节因子。

Mehraj, Umar; Maimekov, Uran; Manzoor, Shaista; Cordova, Emily; Patel, Manasiben; Mancera-Ortiz, Ikeer Y; Howell, Stefanie; Davis-Gilbert, Zachary W; Wang, Mu-En; Chen, Ming; Park, Jung Wook; Wang, Yuzhuo; Armstrong, Andrew J; Huang, Jiaoti; Drewry, David H; Mitrofanova, Antonina; Macias, Everardo

How many kinases are druggable? A review of our current understanding

有多少种激酶是可成药的?对我们目前理解的回顾

Anderson, Brian; Rosston, Peter; Ong, Han Wee; Hossain, Mohammad Anwar; Davis-Gilbert, Zachary W; Drewry, David H

Ethical decision-making climate, moral distress, and intention to leave among ICU professionals in a tertiary academic hospital center

三级教学医院中心重症监护室专业人员的伦理决策氛围、道德困境和离职意愿

Silverman, Henry; Wilson, Tracey; Tisherman, Samuel; Kheirbek, Raya; Mukherjee, Trishna; Tabatabai, Ali; McQuillan, Karen; Hausladen, Rachel; Davis-Gilbert, Melissa; Cho, Eunsung; Bouchard, Kerri; Dove, Samantha; Landon, Julie; Zimmer, Michele

Nuclear Transcriptomes of the Seven Neuronal Cell Types That Constitute the Drosophila Mushroom Bodies

构成果蝇蘑菇体的七种神经元细胞类型的核转录组

Meng-Fu Maxwell Shih, Fred Pejman Davis, Gilbert Lee Henry, Josh Dubnau

Mechanism of Ti-Catalyzed Oxidative Nitrene Transfer in [2 + 2 + 1] Pyrrole Synthesis from Alkynes and Azobenzene

钛催化氧化氮烯转移在炔烃与偶氮苯[2+2+1]吡咯合成中的机理

Davis-Gilbert, Zachary W; Wen, Xuelan; Goodpaster, Jason D; Tonks, Ian A

In Situ Catalyst Generation and Benchtop-Compatible Entry Points for Ti(II)/Ti(IV) Redox Catalytic Reactions

原位催化剂生成及适用于台式操作的Ti(II)/Ti(IV)氧化还原催化反应的入门方法

Davis-Gilbert, Zachary W; Kawakita, Kento; Blechschmidt, Daniel R; Tsurugi, Hayato; Mashima, Kazushi; Tonks, Ian A

Titanium redox catalysis: insights and applications of an earth-abundant base metal

钛氧化还原催化:一种储量丰富的贱金属的见解和应用

Davis-Gilbert, Zachary W; Tonks, Ian A