日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of MK-8353, an orally administered ERK1/2 inhibitor, in patients with advanced solid tumors

口服 ERK1/2 抑制剂 MK-8353 的开发,用于治疗晚期实体肿瘤患者

Stergios J Moschos, Ryan J Sullivan, Wen-Jen Hwu, Ramesh K Ramanathan, Alex A Adjei, Peter C Fong, Ronnie Shapira-Frommer, Hussein A Tawbi, Joseph Rubino, Thomas S Rush 3rd, Da Zhang, Nathan R Miselis, Ahmed A Samatar, Patrick Chun, Eric H Rubin, James Schiller, Brian J Long, Priya Dayananth, Donna

MK-8353: Discovery of an Orally Bioavailable Dual Mechanism ERK Inhibitor for Oncology

MK-8353:一种用于肿瘤治疗的口服生物利用度高的双机制ERK抑制剂的发现

Boga, Sobhana Babu; Deng, Yongqi; Zhu, Liang; Nan, Yang; Cooper, Alan B; Shipps, Gerald W Jr; Doll, Ronald; Shih, Neng-Yang; Zhu, Hugh; Sun, Robert; Wang, Tong; Paliwal, Sunil; Tsui, Hon-Chung; Gao, Xiaolei; Yao, Xin; Desai, Jagdish; Wang, James; Alhassan, Abdul Basit; Kelly, Joseph; Patel, Mehul; Muppalla, Kiran; Gudipati, Subrahmanyam; Zhang, Li-Kang; Buevich, Alexei; Hesk, David; Carr, Donna; Dayananth, Priya; Black, Stuart; Mei, Hong; Cox, Kathleen; Sherborne, Bradley; Hruza, Alan W; Xiao, Li; Jin, Weihong; Long, Brian; Liu, Gongjie; Taylor, Stacey A; Kirschmeier, Paul; Windsor, William T; Bishop, Robert; Samatar, Ahmed A

Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent

基布德洛霉素是一种广谱杀菌剂,可有效对抗需氧菌。

Singh, Sheo B; Dayananth, Priya; Balibar, Carl J; Garlisi, Charles G; Lu, Jun; Kishii, Ryuta; Takei, Masaya; Fukuda, Yasumichi; Ha, Sookhee; Young, Katherine

Discovery of a novel ERK inhibitor with activity in models of acquired resistance to BRAF and MEK inhibitors

发现一种新型 ERK 抑制剂,在 BRAF 和 MEK 抑制剂获得性耐药模型中具有活性

Erick J Morris, Sharda Jha, Clifford R Restaino, Priya Dayananth, Hugh Zhu, Alan Cooper, Donna Carr, Yongi Deng, Weihong Jin, Stuart Black, Brian Long, Jenny Liu, Edward Dinunzio, William Windsor, Rumin Zhang, Shuxia Zhao, Minilik H Angagaw, Elaine M Pinheiro, Jagdish Desai, Li Xiao, Gerald Shipps, 

Analysis of the ERK1,2 transcriptome in mammary epithelial cells

乳腺上皮细胞中ERK1,2转录组的分析

Grill, Constance; Gheyas, Ferdous; Dayananth, Priya; Jin, Weihong; Ding, Wei; Qiu, Ping; Wang, Luquan; Doll, Ronald J; English, Jessie M