日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combined inhibition of NAD synthesis and C-terminal binding protein cooperatively induces cell death and inhibits growth of high grade serous ovarian carcinoma.

NAD 合成和 C 端结合蛋白的联合抑制可协同诱导细胞死亡并抑制高级别浆液性卵巢癌的生长。

Chougoni Kranthi Kumar, West Jacqueline, Martin Nicholette St, Dcona Diana, Kose Istem, Kim Nari, Dcona Martin M, Drapkin Ronny, Carlson Joseph W, Walts Ann E, Orsulic Sandra, Ellis Keith C, Grossman Steven R

Coordinate transcriptional regulation of ErbB2/3 by C-terminal binding protein 2 signals sensitivity to ErbB2 inhibition in pancreatic adenocarcinoma

端结合蛋白 2 对 ErbB2/3 的协调转录调控表明胰腺腺癌对 ErbB2 抑制敏感

Kranthi Kumar Chougoni, Haemin Park, Priyadarshan K Damle, Travis Mason, Bo Cheng, Martin M Dcona, Barbara Szomju, Mikhail G Dozmorov, Michael O Idowu, Steven R Grossman

Combined Targeting of NAD Biosynthesis and the NAD-dependent Transcription Factor C-terminal Binding Protein as a Promising Novel Therapy for Pancreatic Cancer

联合靶向NAD生物合成和NAD依赖性转录因子C端结合蛋白有望成为胰腺癌的一种新型治疗方法

M Michael Dcona ,Kranthi Kumar Chougoni ,Diana T Dcona ,Jacqueline L West ,Sahib J Singh ,Keith C Ellis ,Steven R Grossman

Cryo-EM structure of CtBP2 confirms tetrameric architecture

CtBP2的冷冻电镜结构证实了其四聚体结构

Jecrois, Anne M; Dcona, M Michael; Deng, Xiaoyan; Bandyopadhyay, Dipankar; Grossman, Steven R; Schiffer, Celia A; Royer, William E Jr

Active-Site Tryptophan, the Target of Antineoplastic C-Terminal Binding Protein Inhibitors, Mediates Inhibitor Disruption of CtBP Oligomerization and Transcription Coregulatory Activities

活性位点色氨酸是抗肿瘤C端结合蛋白抑制剂的靶点,它介导抑制剂对CtBP寡聚化和转录共调控活性的破坏。

M Michael Dcona ,Priyadarshan K Damle ,Francisco Zarate-Perez ,Benjamin L Morris ,Zaid Nawaz ,Michael J Dennis ,Xiaoyan Deng ,Sudha Korwar ,Sahib J Singh ,Keith C Ellis ,William E Royer ,Dipankar Bandyopadhyay ,Carlos Escalante ,Steven R Grossman

CtBP- an emerging oncogene and novel small molecule drug target: Advances in the understanding of its oncogenic action and identification of therapeutic inhibitors

CtBP——一种新兴的癌基因和新型小分子药物靶点:对其致癌作用的理解进展及治疗性抑制剂的鉴定

Dcona, M Michael; Morris, Benjamin L; Ellis, Keith C; Grossman, Steven R

Light induced drug release from a folic acid-drug conjugate

光诱导叶酸-药物偶联物释放药物

Dcona, M Michael; Sheldon, Jonathon E; Mitra, Deboleena; Hartman, Matthew C T

Photoswitchable anticancer activity via trans-cis isomerization of a combretastatin A-4 analog

通过康普瑞他汀 A-4 类似物的反式-顺式异构化实现光开关抗癌活性

Jonathon E Sheldon, M Michael Dcona, Charles E Lyons, John C Hackett, Matthew C T Hartman

A new, highly water-soluble, fluorescent turn-on chemodosimeter for direct measurement of hydrogen sulfide in biological fluids

一种新型高水溶性荧光开启型化学剂量计,用于直接测量生物体液中的硫化氢

Hartman, Matthew C T; Dcona, M Michael