日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Complexoform-restricted covalent TRMT112 ligands that allosterically agonize METTL5

具有复合物形式限制的共价TRMT112配体,可变构激动METTL5

Goetzke, F Wieland; Bernard, Steffen M; Ju, Cheng-Wei; Pollock, Jonathan; DeMeester, Kristen E; Gross, Jacob; Simon, Gabriel M; He, Chuan; Melillo, Bruno; Cravatt, Benjamin F

Cysteine Reactivity Profiling Identifies Host Regulators of Mycobacterium tuberculosis Replication in Human Macrophages

半胱氨酸反应性分析揭示人类巨噬细胞中结核分枝杆菌复制的宿主调节因子

Neff, John K; DeMeester, Kristen E; Párraga Solórzano, Paola K; Suciu, Radu M; Dix, Melissa M; Simon, Gabriel; Gianakopoulos, Max A; Melillo, Bruno; Cravatt, Benjamin F; Shiloh, Michael U

Bio-orthogonal Labeling of Chitin in Native Pathogenic Candida Species via the Chitin Scavenge Pathway

通过几丁质清除途径对天然致病性念珠菌物种中的几丁质进行生物正交标记

Williams, Caroline; Carnahan, Bella R; Hyland, Stephen N; DeMeester, Kristen E; Grimes, Catherine L

Complexoform-restricted covalent TRMT112 ligands that allosterically agonize METTL5

具有复合物形式限制的共价TRMT112配体,可变构激动METTL5

Goetzke, F Wieland; Bernard, Steffen M; Ju, Cheng-Wei; Pollock, Jonathan; DeMeester, Kristen E; Gross, Jacob; Simon, Gabriel M; He, Chuan; Melillo, Bruno; Cravatt, Benjamin F

Cysteine reactivity profiling identifies host regulators of Mycobacterium tuberculosis replication in human macrophages

半胱氨酸反应性分析可鉴定人类巨噬细胞中结核分枝杆菌复制的宿主调节因子

Neff, John; DeMeester, Kristen E; Parraga, Paola K; Suciu, Radu; Dix, Melissa; Simon, Gabriel; Gianakopoulos, Max A; Melillo, Bruno; Cravatt, Benjamin F; Shiloh, Michael U

Tryptoline Stereoprobe Elaboration Identifies Inhibitors of the GRPEL1-HSPA9 Chaperone Complex

色氨酸立体探针的衍生化鉴定出 GRPEL1-HSPA9 分子伴侣复合物的抑制剂

Hayward, Rachel E; Berkeley, Raymond F; Gao, Zijian; Garhammer, Maximilian; Morizono, Marc A; Njomen, Evert; Li, Haoxin; DeMeester, Kristen E; Cociorva, Victor; Herzik, Mark A Jr; Hartl, F Ulrich; Melillo, Bruno; Cravatt, Benjamin F

Redirecting the pioneering function of FOXA1 with covalent small molecules.

利用共价小分子重新定向 FOXA1 的先锋功能

Won Sang Joon, Zhang Yuxiang, Reinhardt Christopher J, Hargis Lauren M, MacRae Nicole S, DeMeester Kristen E, Njomen Evert, Remsberg Jarrett R, Melillo Bruno, Cravatt Benjamin F, Erb Michael A

Proteomic Ligandability Maps of Spirocycle Acrylamide Stereoprobes Identify Covalent ERCC3 Degraders

螺环丙烯酰胺立体探针的蛋白质组学配体结合能力图谱鉴定共价ERCC3降解剂

Liu, Zhonglin; Remsberg, Jarrett R; Li, Haoxin; Njomen, Evert; DeMeester, Kristen E; Tao, Yongfeng; Xia, Guoqin; Hayward, Rachel E; Yoo, Minjin; Nguyen, Tracey; Simon, Gabriel M; Schreiber, Stuart L; Melillo, Bruno; Cravatt, Benjamin F

Chemical tools to expand the ligandable proteome: Diversity-oriented synthesis-based photoreactive stereoprobes.

扩展可配体结合蛋白质组的化学工具:基于多样性的合成的光反应立体探针

Ogasawara Daisuke, Konrad David B, Tan Zher Yin, Carey Kimberly L, Luo Jessica, Won Sang Joon, Li Haoxin, Carter Trever R, DeMeester Kristen E, Njomen Evert, Schreiber Stuart L, Xavier Ramnik J, Melillo Bruno, Cravatt Benjamin F

Chemical tools to expand the ligandable proteome: diversity-oriented synthesis-based photoreactive stereoprobes

拓展配体结合蛋白质组的化学工具:基于多样性导向合成的光反应立体探针

Ogasawara, Daisuke; Konrad, David B; Tan, Zher Yin; Carey, Kimberly L; Luo, Jessica; Won, Sang Joon; Li, Haoxin; Carter, Trever; DeMeester, Kristen E; Njomen, Evert; Schreiber, Stuart L; Xavier, Ramnik J; Melillo, Bruno; Cravatt, Benjamin F