日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N-Methyl-D-Aspartate Receptor Hypofunction in Meg-01 Cells Reveals a Role for Intracellular Calcium Homeostasis in Balancing Megakaryocytic-Erythroid Differentiation

Meg-01 细胞中的 N-甲基-D-天冬氨酸受体功能减退揭示了细胞内钙稳态在平衡巨核细胞-红细胞分化中的作用

James I Hearn, Taryn N Green, Martin Chopra, Yohanes N S Nursalim, Leandro Ladvanszky, Nicholas Knowlton, Cherie Blenkiron, Raewyn C Poulsen, Dean C Singleton, Stefan K Bohlander, Maggie L Kalev-Zylinska

Pyruvate anaplerosis is a mechanism of resistance to pharmacological glutaminase inhibition in triple-receptor negative breast cancer

丙酮酸补充是三受体阴性乳腺癌对药物谷氨酰胺酶抑制产生抵抗的机制

Dean C Singleton, Anne-Lise Dechaume, Pamela M Murray, William P Katt, Bruce C Baguley, Euphemia Y Leung

Derivation of Breast Cancer Cell Lines Under Physiological (5%) Oxygen Concentrations

生理(5%)氧气浓度下乳腺癌细胞系的衍生

Euphemia Y Leung, Marjan E Askarian-Amiri, Dean C Singleton, Carole Ferraro-Peyret, Wayne R Joseph, Graeme J Finlay, Reuben J Broom, Purvi M Kakadia, Stefan K Bohlander, Elaine Marshall, Bruce C Baguley

LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor

LP99:首个选择性 BRD7/9 溴结构域抑制剂的发现和合成

Peter G K Clark, Lucas C C Vieira, Cynthia Tallant, Oleg Fedorov, Dean C Singleton, Catherine M Rogers, Octovia P Monteiro, James M Bennett, Roberta Baronio, Susanne Müller, Danette L Daniels, Jacqui Méndez, Stefan Knapp, Paul E Brennan, Darren J Dixon

Discovery and optimization of small-molecule ligands for the CBP/p300 bromodomains

CBP/p300 溴结构域小分子配体的发现和优化

Duncan A Hay, Oleg Fedorov, Sarah Martin, Dean C Singleton, Cynthia Tallant, Christopher Wells, Sarah Picaud, Martin Philpott, Octovia P Monteiro, Catherine M Rogers, Stuart J Conway, Timothy P C Rooney, Anthony Tumber, Clarence Yapp, Panagis Filippakopoulos, Mark E Bunnage, Susanne Müller, Stefan K