日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of mCMV280: An Oral Ectoparasiticide in the Isoxazoline Class with Reduced Mammalian Brain Exposure

mCMV280 的发现:一种异噁唑啉类口服体外寄生虫杀灭剂,可降低哺乳动物大脑暴露量

McComic, Sarah E; Wilson, Katy B; Li, Zhilin; Chen, Jeffrey; Weiss, Frank; Song, Lirui; Mazumdar, Wrickban; Dvorak, Curt A; Brittain, Jason; Lee, Kyoung-Jin; Li, Shuangwei; Joseph, Sean B; McNamara, Case W; Vos, Martijn W; Sheshachalam, Avinash; Inácio, Alex; Dechering, Koen J; Chatterjee, Arnab K; Swale, Daniel R

The kinetics and transmission-blocking dynamics of P. falciparum sexual-stage antibody responses in a six-year cohort of Ugandan children and adults

乌干达儿童和成人六年队列研究中恶性疟原虫性阶段抗体反应的动力学和阻断传播动态

Blanken, Sara Lynn; Nayebare, Patience; Briese, Jonathan; Nijman, Gerine; Teelen, Karina; Stoter, Rianne; van Gemert, Geert-Jan; Graumans, Wouter; Oulton, Tate; Patterson, Catriona; Drammeh, Abdoulie; de Bruijni, Marloes; Bolscher, Judith; Cohee, Lauren M; Kumar, Sanjai; Sather, Noah; Molina-Cruz, Alvaro; Arinaitwe, Emmanuel; Kamya, Moses R; Dechering, Koen; Dorsey, Grant; Drakeley, Chris; Jore, Matthijs M; Bousema, Teun; Stone, William

Temperature to time Catch-Up: a novel procedural endpoint to predict durable pulmonary vein isolation after cryoballoon ablation of paroxysmal atrial fibrillation

温度-时间追赶:一种预测阵发性房颤冷冻球囊消融术后持久肺静脉隔离的新型手术终点

Willy, Kevin; Wolfes, Julian; Müller, Patrick; Ellermann, Christian; Dechering, Dirk; Lange, Philipp S; Rath, Benjamin; Reinke, Florian; Doldi, Florian; Güner, Fatih; Köbe, Julia; Leitz, Patrick; Frommeyer, Gerrit; Laredo, Mikael; Eckardt, Lars

An accessible 3D HepG2/C3A liver spheroid model supporting the complete intrahepatocytic lifecycle of Plasmodium falciparum.

一种易于操作的 3D HepG2/C3A 肝球体模型,支持恶性疟原虫完整的肝细胞内生命周期。

Caygill Claire H, Alqurashi Salwa Omar, Adolfi Adriana, Carson Jessica, Sturm Angelika, Evans Daniel S, Jinks Jess B, Dechering Koen J, Reimer Lisa, Pennington Shaun H, Sharma Parveen, Ward Stephen A, Biagini Giancarlo A

A deep learning and digital archaeology approach for mosquito repellent discovery

利用深度学习和数字考古学方法发现驱蚊剂

Wei, Jennifer N; Ruiz, Carlos; Vlot, Marnix; Sanchez-Lengeling, Benjamin; Lee, Brian K; Berning, Luuk; Vos, Martijn W; Henderson, Rob W M; Qian, Wesley W; Sanders, Jacob N; Ando, D Michael; Groetsch, Kurt M; Gerkin, Richard C; Wiltschko, Alexander B; Riffell, Jeffrey A; Dechering, Koen J

Revisiting the Plasmodium falciparum druggable genome using predicted structures and data mining

利用预测结构和数据挖掘技术重新审视恶性疟原虫可药物靶向基因组

Godinez-Macias, Karla P; Chen, Daisy; Wallis, J Lincoln; Siegel, Miles G; Adam, Anna; Bopp, Selina; Carolino, Krypton; Coulson, Lauren B; Durst, Greg; Thathy, Vandana; Esherick, Lisl; Farringer, Madeline A; Flannery, Erika L; Forte, Barbara; Liu, Tiqing; Godoy Magalhaes, Luma; Gupta, Anil K; Istvan, Eva S; Jiang, Tiantian; Kumpornsin, Krittikorn; Lobb, Karen; McLean, Kyle J; Moura, Igor M R; Okombo, John; Payne, N Connor; Plater, Andrew; Rao, Srinivasa P S; Siqueira-Neto, Jair L; Somsen, Bente A; Summers, Robert L; Zhang, Rumin; Gilson, Michael K; Gamo, Francisco-Javier; Campo, Brice; Baragaña, Beatriz; Duffy, James; Gilbert, Ian H; Lukens, Amanda K; Dechering, Koen J; Niles, Jacquin C; McNamara, Case W; Cheng, Xiu; Birkholtz, Lyn-Marie; Bronkhorst, Alfred W; Fidock, David A; Wirth, Dyann F; Goldberg, Daniel E; Lee, Marcus C S; Winzeler, Elizabeth A

Inhibitors of malaria parasite cyclic nucleotide phosphodiesterases block asexual blood-stage development and mosquito transmission.

疟原虫环核苷酸磷酸二酯酶抑制剂可阻断无性血液期发育和蚊子传播

Gomez-Gonzalez Paula-Josefina, Gupta Antima, Drought Laura G, Patel Avnish, Okombo John, van der Watt Mariëtte, Walker-Gray Ryan, Schindler Kyra A, Burkhard Anna Y, Yeo Tomas, Narwal Sunil K, Bloxham Talia S, Flueck Christian, Walker Eloise M, Rey Joshua A, Fairhurst Kate J, Reader Janette, Park Heekuk, Pollard Harry G, Stewart Lindsay B, Brandner-Garrod Luke, Kristan Mojca, Sterk Geert-Jan, van Nuland Youri M, Manko Emilia, van Schalkwyk Donelly A, Zheng Yang, Leurs Rob, Dechering Koen J, Aguiar Anna Caroline C, Guido Rafael V C, Pereira Dhelio B, Tumwebaze Patrick K, Nosbya Samuel L, Rosenthal Philip J, Cooper Roland A, Palmer Mike, Parkinson Tanya, Burrows Jeremy N, Uhlemann Anne-Catrin, Birkholtz Lyn-Marié, Small-Saunders Jennifer L, Duffy James, Fidock David A, Brown Alan, Gardner Mark, Baker David A

Revisiting the Plasmodium falciparum druggable genome using predicted structures and data mining

利用预测结构和数据挖掘技术重新审视恶性疟原虫可药物靶向基因组

Godinez-Macias, Karla P; Chen, Daisy; Wallis, J Lincoln; Siegel, Miles G; Adam, Anna; Bopp, Selina; Carolino, Krypton; Coulson, Lauren B; Durst, Greg; Thathy, Vandana; Esherick, Lisl; Farringer, Madeline A; Flannery, Erika L; Forte, Barbara; Liu, Tiqing; Magalhaes, Luma Godoy; Gupta, Anil K; Istvan, Eva S; Jiang, Tiantian; Kumpornsin, Krittikorn; Lobb, Karen; McLean, Kyle; Moura, Igor M R; Okombo, John; Payne, N Connor; Plater, Andrew; Rao, Srinivasa P S; Siqueira-Neto, Jair L; Somsen, Bente A; Summers, Robert L; Zhang, Rumin; Gilson, Michael K; Gamo, Francisco-Javier; Campo, Brice; Baragaña, Beatriz; Duffy, James; Gilbert, Ian H; Lukens, Amanda K; Dechering, Koen J; Niles, Jacquin C; McNamara, Case W; Cheng, Xiu; Birkholtz, Lyn-Marie; Bronkhorst, Alfred W; Fidock, David A; Wirth, Dyann F; Goldberg, Daniel E; Lee, Marcus C S; Winzeler, Elizabeth A

Highly potent, naturally acquired human monoclonal antibodies against Pfs48/45 block Plasmodium falciparum transmission to mosquitoes

针对Pfs48/45的高效天然人单克隆抗体可阻断恶性疟原虫向蚊子的传播。

Amanda Fabra-García ,Sophia Hailemariam ,Roos M de Jong ,Kirsten Janssen ,Karina Teelen ,Marga van de Vegte-Bolmer ,Geert-Jan van Gemert ,Danton Ivanochko ,Anthony Semesi ,Brandon McLeod ,Martijn W Vos ,Marloes H C de Bruijni ,Judith M Bolscher ,Marta Szabat ,Stefanie Vogt ,Lucas Kraft ,Sherie Duncan ,Moses R Kamya ,Margaret E Feeney ,Prasanna Jagannathan ,Bryan Greenhouse ,Koen J Dechering ,Robert W Sauerwein ,C Richter King ,Randall S MacGill ,Teun Bousema ,Jean-Philippe Julien ,Matthijs M Jore

Metabolic activity organizes olfactory representations

代谢活动组织嗅觉表征

Qian, Wesley W; Wei, Jennifer N; Sanchez-Lengeling, Benjamin; Lee, Brian K; Luo, Yunan; Vlot, Marnix; Dechering, Koen; Peng, Jian; Gerkin, Richard C; Wiltschko, Alexander B