Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice
通过先导优化筛选高亲和力、变构细胞周期蛋白依赖性激酶 2 (CDK2) 抑制剂作为减少小鼠精子数量的男性避孕药
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c01731
Erik B Faber, Nan Wang, Kristen John, Luxin Sun, Henry L Wong, David Burban, Rawle Francis, Defeng Tian, Kwon H Hong, An Yang, Liming Wang, Mazen Elsaid, Hira Khalid, Nicholas M Levinson, Ernst Schönbrunn, Jon E Hawkinson, Gunda I Georg