日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PepFuNN: Novo Nordisk Open-Source Toolkit to Enable Peptide in Silico Analysis

PepFuNN:诺和诺德开源工具包,用于实现肽的计算机模拟分析

Ochoa, Rodrigo; Deibler, Kristine

De novo design of miniprotein agonists and antagonists targeting G protein-coupled receptors.

从头设计靶向 G 蛋白偶联受体的微型蛋白激动剂和拮抗剂

Muratspahić Edin, Feldman David, Kim David E, Qu Xiangli, Bratovianu Ana-Maria, Rivera-Sánchez Paula, Dimitri Federica, Cao Jason, Cary Brian P, Belousoff Matthew J, Keov Peter, Chen Qingchao, Ren Yue, Fine Justyn, Sappington Isaac, Schlichthaerle Thomas, Zhang Jason Z, Pillai Arvind, Mihaljević Ljubica, Bauer Magnus, Torres Susana Vázquez, Motmaen Amir, Lee Gyu Rie, Tran Long, Wang Xinru, Goreshnik Inna, Vafeados Dionne K, Svendsen Justin E, Hosseinzadeh Parisa, Lindegaard Nicolai, Brandt Matthäus, Waltenspühl Yann, Deibler Kristine, Oostdyk Luke, Cao William, Anantharaman Lakshmi, Stewart Lance, Halloran Lauren, Spangler Jamie B, Sexton Patrick M, Roth Bryan L, Krumm Brian E, Wootten Denise, Tate Christopher G, Norn Christoffer, Baker David

Glp1r-Lepr coexpressing neurons modulate the suppression of food intake and body weight by a GLP-1/leptin dual agonist

共表达 Glp1r-Lepr 的神经元通过 GLP-1/瘦素双重激动剂调节食物摄入和体重的抑制。

Polex-Wolf, Joseph; Deibler, Kristine; Hogendorf, Wouter Frederik Johan; Bau, Sarah; Glendorf, Tine; Stidsen, Carsten Enggaard; Tornøe, Christian Wenzel; Tiantang, Dong; Lundh, Sofia; Pyke, Charles; Tomlinson, Abigail J; Kernodle, Stace; Magrisso, Irwin Jack; Conde-Frieboes, Kilian W; Myers, Martin G Jr; Knudsen, Lotte Bjerre; Seeley, Randy J

Rational Design of Highly Potent and Selective Covalent MAP2K7 Inhibitors

高效选择性共价MAP2K7抑制剂的合理设计

Kim, Dalton R; Orr, Meghan J; Kwong, Ada J; Deibler, Kristine K; Munshi, Hasan H; Bridges, Cory Seth; Chen, Taylor Jie; Zhang, Xiaoyu; Lacorazza, H Daniel; Scheidt, Karl A

An integrated platform approach enables discovery of potent, selective and ligand-competitive cyclic peptides targeting the GIP receptor

整合平台方法能够发现靶向GIP受体的高效、选择性强且具有配体竞争性的环状肽。

Bhushan, Bhaskar; Granata, Daniele; Kaas, Christian S; Kasimova, Marina A; Ren, Qiansheng; Cramer, Christian N; White, Mark D; Hansen, Ann Maria K; Fledelius, Christian; Invernizzi, Gaetano; Deibler, Kristine; Coleman, Oliver D; Zhao, Xin; Qu, Xinping; Liu, Haimo; Zurmühl, Silvana S; Kodra, Janos T; Kawamura, Akane; Münzel, Martin

A79 CHARACTERISTICS OF PEDIATRIC INFLAMMATORY BOWEL DISEASE AT DIAGNOSIS RELATED TO EARLIER USE OF BIOLOGIC THERAPY

A79 早期生物疗法对儿童炎症性肠病诊断特征的影响

Thomas, Nidhin; Sanyal, Tanmoy; Greisen, Per Jr; Deibler, Kristine; Mulder, D J; Zachos, M; Issenman, R; Sherlock, M

Synthesis and Biological Evaluation of 3-Arylindazoles as Selective MEK4 Inhibitors

3-芳基吲唑类化合物作为选择性MEK4抑制剂的合成及生物学评价

Deibler, Kristine K; Schiltz, Gary E; Clutter, Matthew R; Mishra, Rama K; Vagadia, Purav P; O'Connor, Matthew; George, Mariam Donny; Gordon, Ryan; Fowler, Graham; Bergan, Raymond; Scheidt, Karl A