日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Crystallographic characterisation and development of bi-substrate inhibitors of coronavirus nsp14 methyltransferase

冠状病毒nsp14甲基转移酶双底物抑制剂的晶体学表征和开发

Georgiou, Irene; Robinson, Colin; O'Byrne, Sean N; Matsuda, Alex; Grygier, Przemysław; Smith, Craig D; O'Neill, Sandra; Ahmad, Shamshad A; Norval, Suzanne; Post, John M; Groenewold, Mirjam; Urakova, Nadya; Wanningen, Patrick; Kresik, Leanid; Plewka, Jacek; Delpal, Adrien; See, Kexin; Eadsforth, Thomas; Wierzbicka, Kinga; Decroly, Etienne; Saikatendu, Kumar Singh; Chang, Edcon; Snijder, Eric J; Pyrć, Krzysztof; Czarna, Anna; Scott, Duncan E; Gilbert, Ian H

N-Arylsulfonamide-based adenosine analogues to target RNA cap N7-methyltransferase nsp14 of SARS-CoV-2

基于N-芳基磺酰胺的腺苷类似物靶向SARS-CoV-2的RNA帽N7-甲基转移酶nsp14

Ahmed-Belkacem, Rostom; Troussier, Joris; Delpal, Adrien; Canard, Bruno; Vasseur, Jean-Jacques; Decroly, Etienne; Debart, Françoise

Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases

腺苷类似物的结构引导优化作为冠状病毒 nsp14 N7-甲基转移酶的选择性和有效抑制剂

Marcel Hausdorff, Adrien Delpal, Sarah Barelier, Laura Nicollet, Bruno Canard, Franck Touret, Agathe Colmant, Bruno Coutard, Jean-Jacques Vasseur, Etienne Decroly, Françoise Debart

Design and synthesis of naturally-inspired SARS-CoV-2 inhibitors

天然SARS-CoV-2抑制剂的设计与合成

Hassan, Haitham; Chiavaralli, Jeanne; Hassan, Afnan; Bedda, Loay; Krischuns, Tim; Chen, Kuang-Yu; Li, Alice Shi Ming; Delpal, Adrien; Decroly, Etienne; Vedadi, Masoud; Naffakh, Nadia; Agou, Fabrice; Mallart, Sergio; Arafa, Reem K; Arimondo, Paola B

Synthesis, Structure-Activity Relationships, and Antiviral Profiling of 1-Heteroaryl-2-Alkoxyphenyl Analogs as Inhibitors of SARS-CoV-2 Replication

1-杂芳基-2-烷氧基苯基类似物作为 SARS-CoV-2 复制抑制剂的合成、构效关系和抗病毒分析

Dorothée Bardiot, Laura Vangeel, Mohamed Koukni, Philippe Arzel, Marleen Zwaagstra, Heyrhyoung Lyoo, Patrick Wanningen, Shamshad Ahmad, Linlin Zhang, Xinyuanyuan Sun, Adrien Delpal, Cecilia Eydoux, Jean-Claude Guillemot, Eveline Lescrinier, Hugo Klaassen, Pieter Leyssen, Dirk Jochmans, Karolien Cast

Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity

Furin 和 TMPRSS2 在 SARS-CoV-2 传染性中的独特作用

Rachid Essalmani, Jaspreet Jain #, Delia Susan-Resiga #, Ursula Andréo #, Alexandra Evagelidis, Rabeb Mouna Derbali, David N Huynh, Frédéric Dallaire, Mélanie Laporte, Adrien Delpal, Priscila Sutto-Ortiz, Bruno Coutard, Claudine Mapa, Keith Wilcoxen, Etienne Decroly, Tram Nq Pham, Éric A Cohen, Nabi

Erratum for Essalmani et al., "Distinctive Roles of Furin and TMPRSS2 in SARS-CoV-2 Infectivity"

Essalmani 等人的论文“Furin 和 TMPRSS2 在 SARS-CoV-2 感染性中的独特作用”的勘误

Essalmani, Rachid; Jain, Jaspreet; Susan-Resiga, Delia; Andréo, Ursula; Evagelidis, Alexandra; Derbali, Rabeb Mouna; Huynh, David N; Dallaire, Frédéric; Laporte, Mélanie; Delpal, Adrien; Sutto-Ortiz, Priscila; Coutard, Bruno; Mapa, Claudine; Wilcoxen, Keith; Decroly, Etienne; Pham, Tram N Q; Cohen, Éric A; Seidah, Nabil G

A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro

一类用途广泛的 1,4,4-三取代哌啶类化合物可在体外阻断冠状病毒复制

Sonia De Castro, Annelies Stevaert, Miguel Maldonado, Adrien Delpal, Julie Vandeput, Benjamin Van Loy, Cecilia Eydoux, Jean-Claude Guillemot, Etienne Decroly, Federico Gago, Bruno Canard, Maria-Jose Camarasa, Sonsoles Velázquez, Lieve Naesens

Oxytocin stimulates secretory processes in lactating rabbit mammary epithelial cells

催产素刺激哺乳期兔乳腺上皮细胞的分泌过程。

Lollivier, Vanessa; Marnet, Pierre-Guy; Delpal, Serge; Rainteau, Dominique; Achard, Caroline; Rabot, Aline; Ollivier-Bousquet, Michèle