Optimization of Brain Penetrant SARM1 Orthosteric Inhibitors and Discovery of Their Paradoxical Subinhibitory Activation
优化脑穿透性SARM1正构抑制剂及其矛盾的亚抑制激活作用
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00189
Green, Samantha A; Smith, Russell T; Grandner, Jessica M; Zeng, Mingshuo; Del Bel, Matthew; Zhu, Bing-Yan; Liang, Jun; Braun, Marie-Gabrielle; Sudhamsu, Jawahar; Wallweber, Heidi Ackerly; Boenig, Gladys; Murray, Jeremy; Shen, Xiaoli; Zhang, Renwei; Lai, Kwong Wah; Delwig, Anton; Breboneria, Maria Andrea; Ly, Justin; Ganti, Anjani; Nespi, Marika; Weber, Martin; Leahey, Rebecca; Hinz, Flora I; Chan, Bryan K