日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evidence for the Quercetin Binding Site of Glycogen Phosphorylase as a Target for Liver-Isoform-Selective Inhibitors against Glioblastoma: Investigation of Flavanols Epigallocatechin Gallate and Epigallocatechin

槲皮素结合位点作为肝亚型选择性抑制剂治疗胶质母细胞瘤的靶点的证据:表没食子儿茶素没食子酸酯和表没食子儿茶素的研究

Alexopoulos, Serafeim; McGawley, Megan; Mathews, Roshini; Papakostopoulou, Souzana; Koulas, Symeon; Leonidas, Demetres D; Zwain, Tamara; Hayes, Joseph M; Skamnaki, Vasiliki

Kinetic and Structural Studies of the Plastidial Solanum tuberosum Phosphorylase

马铃薯质体磷酸化酶的动力学和结构研究

Koulas, Symeon M; Kyriakis, Efthimios; Tsagkarakou, Anastasia S; Leonidas, Demetres D

Silver ciprofloxacin (CIPAG): a multitargeted metallodrug in the development of breast cancer therapy

银环丙沙星(CIPAG):一种用于乳腺癌治疗的多靶点金属药物

Christina N Banti, Foteini D Kalousi, Anna-Maria G Psarra, Eleni E Moushi, Demetres D Leonidas, Sotiris K Hadjikakou

Biochemical and in silico identification of the active site and the catalytic mechanism of the circadian deadenylase HESPERIN

昼夜节律脱腺苷酸酶 HESPERIN 的活性位点和催化机制的生化和计算机识别

Rafailia A A Beta, Athanasios Kyritsis, Veroniki Douka, Eirini Papanastasi, Marianna Rizouli, Demetres D Leonidas, Dimitrios Vlachakis, Nikolaos A A Balatsos

Glycogen phosphorylase revisited: extending the resolution of the R- and T-state structures of the free enzyme and in complex with allosteric activators

糖原磷酸化酶研究进展:进一步解析游离酶及其与变构激活剂复合物的R态和T态结构

Leonidas, Demetres D; Zographos, Spyros E; Tsitsanou, Katerina E; Skamnaki, Vassiliki T; Stravodimos, George; Kyriakis, Efthimios

Nicotinic cholinergic system and COVID-19: In silico evaluation of nicotinic acetylcholine receptor agonists as potential therapeutic interventions

尼古丁胆碱能系统与新冠肺炎:尼古丁乙酰胆碱受体激动剂作为潜在治疗干预措施的计算机模拟评估

Alexandris, Nikolaos; Lagoumintzis, George; Chasapis, Christos T; Leonidas, Demetres D; Papadopoulos, Georgios E; Tzartos, Socrates J; Tsatsakis, Aristidis; Eliopoulos, Elias; Poulas, Konstantinos; Farsalinos, Konstantinos

Nicotinic Cholinergic System and COVID-19: In Silico Identification of an Interaction between SARS-CoV-2 and Nicotinic Receptors with Potential Therapeutic Targeting Implications

尼古丁胆碱能系统与新冠病毒:计算机模拟鉴定SARS-CoV-2与尼古丁受体之间的相互作用及其潜在的治疗靶点意义

Farsalinos, Konstantinos; Eliopoulos, Elias; Leonidas, Demetres D; Papadopoulos, Georgios E; Tzartos, Socrates; Poulas, Konstantinos

High Consistency of Structure-Based Design and X-Ray Crystallography: Design, Synthesis, Kinetic Evaluation and Crystallographic Binding Mode Determination of Biphenyl- N-acyl-β-d-Glucopyranosylamines as Glycogen Phosphorylase Inhibitors

基于结构的设计与X射线晶体学的高度一致性:联苯-N-酰基-β-d-葡萄吡喃胺作为糖原磷酸化酶抑制剂的设计、合成、动力学评估和晶体学结合模式测定

Thomas Fischer, Symeon M Koulas, Anastasia S Tsagkarakou, Efthimios Kyriakis, George A Stravodimos, Vassiliki T Skamnaki, Panagiota G V Liggri, Spyros E Zographos, Rainer Riedl, Demetres D Leonidas1

Oxidation of human serum albumin exhibits inter-individual variability after an ultra-marathon mountain race

超级马拉松山地赛后,人血清白蛋白的氧化程度表现出个体差异。

Spanidis, Ypatios; Priftis, Alexandros; Stagos, Dimitrios; Stravodimos, George A; Leonidas, Demetres D; Spandidos, Demetrios A; Tsatsakis, Aristides M; Kouretas, Demetrios

AtHESPERIN: a novel regulator of circadian rhythms with poly(A)-degrading activity in plants

AtHESPERIN:一种具有植物中 poly(A) 降解活性的新型昼夜节律调节剂

Costas Delis, Afrodite Krokida, Anastasia Tomatsidou, Daniela Tsikou, Rafailia A A Beta, Maria Tsioumpekou, Julietta Moustaka, Georgios Stravodimos, Demetres D Leonidas, Nikolaos A A Balatsos, Kalliope K Papadopoulou