A biphenyl inhibitor of eIF4E targeting an internal binding site enables the design of cell-permeable PROTAC-degraders
一种靶向eIF4E内部结合位点的联苯抑制剂可用于设计细胞可渗透的PROTAC降解剂。
期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2021.113435
Fischer, Patrick D; Papadopoulos, Evangelos; Dempersmier, Jon M; Wang, Zi-Fu; Nowak, Radosław P; Donovan, Katherine A; Kalabathula, Joann; Gorgulla, Christoph; Junghanns, Pierre P M; Kabha, Eihab; Dimitrakakis, Nikolaos; Petrov, Ognyan I; Mitsiades, Constantine; Ducho, Christian; Gelev, Vladimir; Fischer, Eric S; Wagner, Gerhard; Arthanari, Haribabu