日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Safety, pharmacokinetic, pharmacodynamic, and efficacy properties of orally administered APG-2449 in patients with advanced ALK (+) and ROS1 (+) non-small-cell lung cancer: a multicentre, open-label, single-arm phase 1 trial

口服APG-2449治疗晚期ALK(+)和ROS1(+)非小细胞肺癌患者的安全性、药代动力学、药效学和疗效:一项多中心、开放标签、单臂I期试验

Ma, Yuxiang; Song, Zhengbo; Chen, Jianhua; Zhao, Yanqiu; Fang, Wenfeng; Guo, Yubiao; Dong, Yugang; Yang, Yunpeng; Wu, Gang; Fang, Jian; Lin, Xiaoyan; Li, Jundong; Huang, Yan; Zhao, Yuanyuan; Hong, Shaodong; Xue, Jinhui; Zhang, Yang; Liu, Qianwen; Yang, Chen; Xu, Liang; Yang, Yun; Xiong, Dengkun; Yang, Dajun; Zhai, Yifan; Zhang, Li; Zhao, Hongyun

Effects of the plant growth-promoting rhizobacterium Zobellella sp. DQSA1 on alleviating salt-alkali stress in job's tears seedings and its growth-promoting mechanism

植物促生根际细菌 Zobellella sp. DQSA1 对缓解薏苡幼苗盐碱胁迫的影响及其促生机制

Li, Youzhen; Huang, Yulan; Ding, Hongxia; Huang, Yibo; Xu, Dengkun; Zhan, Shihan; Ma, Mingli

Xixin Decoction's novel mechanism for alleviating Alzheimer's disease cognitive dysfunction by modulating amyloid-β transport across the blood-brain barrier to reduce neuroinflammation

细辛汤通过调节β淀粉样蛋白跨血脑屏障运输以减少神经炎症,减轻阿尔茨海默病认知功能障碍的新机制

Chaokai Yang #, Enlong Zhao, Hu Zhang, Liqi Duan, Xinyue Han, Hongli Ding, Yan Cheng, Dengkun Wang, Xiaojing Lei, Yongchang Diwu #

Risk factors and traditional Chinese medicine syndromes of mild cognitive impairment in community-dwelling hypertensive older adults

社区居住的高血压老年人轻度认知障碍的危险因素和中医证候

Gao, Jie; Wu, Meirong; Jia, Siyuan; Tian, Yuan; Wang, Dengkun; Lei, Xiaojing; Diwu, Yongchang

Discovery of a novel ALK/ROS1/FAK inhibitor, APG-2449, in preclinical non-small cell lung cancer and ovarian cancer models

在临床前非小细胞肺癌和卵巢癌模型中发现新型 ALK/ROS1/FAK 抑制剂 APG-2449

Douglas D Fang #, Ran Tao #, Guangfeng Wang, Yuanbao Li, Kaixiang Zhang, Chunhua Xu, Guoqin Zhai, Qixin Wang, Jingwen Wang, Chunyang Tang, Ping Min, Dengkun Xiong, Jianyong Chen, Shaomeng Wang #, Dajun Yang #, Yifan Zhai #

MicroRNA-432 is downregulated in osteosarcoma and inhibits cell proliferation and invasion by directly targeting metastasis-associated in colon cancer-1

MicroRNA-432在骨肉瘤中表达下调,并通过直接靶向结肠癌转移相关蛋白-1抑制细胞增殖和侵袭。

Lv, Dengkun; Zhen, Zhen; Huang, Defa

MDM2 inhibitor APG-115 exerts potent antitumor activity and synergizes with standard-of-care agents in preclinical acute myeloid leukemia models

MDM2 抑制剂 APG-115 在临床前急性髓系白血病模型中发挥强大的抗肿瘤活性并与标准治疗药物产生协同作用

Douglas D Fang #, Qiuqiong Tang #, Yanhui Kong, Tao Rong, Qixin Wang, Na Li, Xu Fang, Jiaxing Gu, Dengkun Xiong, Yan Yin, Jing Deng, Dajun Yang, Yifan Zhai

MicroRNA-432 is downregulated in osteosarcoma and inhibits cell proliferation and invasion by directly targeting metastasis-associated in colon cancer-1

MicroRNA-432 在骨肉瘤中下调,并通过直接靶向结肠癌转移相关基因-1 来抑制细胞增殖和侵袭

Dengkun Lv, Zhen Zhen, Defa Huang

Oct4 regulates DNA methyltransferase 1 transcription by direct binding of the regulatory element

Oct4 通过直接结合调控元件来调节 DNA 甲基转移酶 1 的转录

Fengrui Wu, Qingqing Wu, Dengkun Li, Yuan Zhang, Rong Wang, Yong Liu, Wenyong Li

Supplement of Betaine into Embryo Culture Medium Can Rescue Injury Effect of Ethanol on Mouse Embryo Development.

在胚胎培养基中添加甜菜碱可以挽救乙醇对小鼠胚胎发育的损伤作用

Zhang Di, Jing Huaijiang, Dou Changfeng, Zhang Ling, Wu Xiaoqing, Wu Qingqing, Song Haoyang, Li Dengkun, Wu Fengrui, Liu Yong, Li Wenyong, Wang Rong