日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Excelsatoxin A-Receptor TMEM233 Modulates Nav1.8

Excelsatoxin A 受体 TMEM233 调节 Nav1.8

Oprita, George; Meyer, Marvin J A; Rudolf, Daniel; Pombeiro Stein, Inês C A; Deuis, Jennifer R; Tran, Hue N T; Durek, Thomas; Tabea, Klasfauseweh; Sina, Jami; Waxman, Stephen G; Dib-Hajj, Sulayman D; Babes, Alexandru; Vetter, Irina; Leffler, Andreas

Refining the Na(V)1.7 pharmacophore of a class of venom-derived peptide inhibitors via a combination of in silico screening and rational engineering

通过计算机筛选和合理设计相结合的方法,优化一类毒液衍生肽抑制剂的Na(V)1.7药效团。

Sharma, Gagan; Deuis, Jennifer R; Jia, Xinying; Crawford, Theo; Rahnama, Sassan; Undheim, Eivind A B; Vetter, Irina; Chin, Yanni K-Y; Mobli, Mehdi

Structural Basis of the Bivalency of the TRPV1 Agonist DkTx

TRPV1激动剂DkTx双价性的结构基础

Ramanujam, Venkatraman; Crawford, Theo; Cristofori-Armstrong, Ben; Deuis, Jennifer R; Jia, Xinying; Maxwell, Michael J; Jami, Sina; Ma, Linlin; Vetter, Irina; Mobli, Mehdi

A venom peptide-induced Na(V) channel modulation mechanism involving the interplay between fixed channel charges and ionic gradients

毒液肽诱导的Na(V)通道调节机制涉及固定通道电荷和离子梯度之间的相互作用

Thapa, Ashvriya; Beh, Jia Hao; Robinson, Samuel D; Deuis, Jennifer R; Tran, Hue; Vetter, Irina; Keramidas, Angelo

Peptide toxins that target vertebrate voltage-gated sodium channels underly the painful stings of harvester ants

收获蚁蜇刺疼痛的根本原因在于其毒素是靶向脊椎动物电压门控钠通道的肽类毒素。

Robinson, Samuel D; Deuis, Jennifer R; Niu, Pancong; Touchard, Axel; Mueller, Alexander; Schendel, Vanessa; Brinkwirth, Nina; King, Glenn F; Vetter, Irina; Schmidt, Justin O

Erythromelalgia caused by the missense mutation p.Arg220Pro in an alternatively spliced exon of SCN9A (NaV1.7)

由 SCN9A (NaV1.7) 的可变剪接外显子中的错义突变 p.Arg220Pro 引起的红斑性肢痛症

Jennifer R Deuis, Smitha Kumble, Angelo Keramidas, Lotten Ragnarsson, Cas Simons, Lynn Pais, Susan M White, Irina Vetter

Ant venoms contain vertebrate-selective pain-causing sodium channel toxins

蚂蚁毒液中含有对脊椎动物具有选择性的、可引起疼痛的钠通道毒素。

Robinson, Samuel D; Deuis, Jennifer R; Touchard, Axel; Keramidas, Angelo; Mueller, Alexander; Schroeder, Christina I; Barassé, Valentine; Walker, Andrew A; Brinkwirth, Nina; Jami, Sina; Bonnafé, Elsa; Treilhou, Michel; Undheim, Eivind A B; Schmidt, Justin O; King, Glenn F; Vetter, Irina

Pain-causing stinging nettle toxins target TMEM233 to modulate NaV1.7 function

引起疼痛的荨麻毒素靶向 TMEM233 来调节 NaV1.7 功能

Sina Jami #, Jennifer R Deuis #, Tabea Klasfauseweh #, Xiaoyang Cheng, Sergey Kurdyukov, Felicity Chung, Andrei L Okorokov, Shengnan Li, Jiangtao Zhang, Ben Cristofori-Armstrong, Mathilde R Israel, Robert J Ju, Samuel D Robinson, Peng Zhao, Lotten Ragnarsson, Åsa Andersson, Poanna Tran, Vanessa Sche

Identification of sodium channel toxins from marine cone snails of the subgenera Textilia and Afonsoconus

从海洋锥螺亚属 Textilia 和 Afonsoconus 中鉴定钠通道毒素

McMahon, Kirsten L; O'Brien, Henrik; Schroeder, Christina I; Deuis, Jennifer R; Venkatachalam, Dhananjeyan; Huang, Di; Green, Brad R; Bandyopadhyay, Pradip K; Li, Qing; Yandell, Mark; Safavi-Hemami, Helena; Olivera, Baldomero M; Vetter, Irina; Robinson, Samuel D

Natural Compounds Purified from the Leaves of Aristotelia chilensis: Makomakinol, a New Alkaloid and the Effect of Aristoteline and Hobartine on Na(V) Channels

从智利马兜铃叶中纯化的天然化合物:一种新的生物碱马可马金醇以及马兜铃碱和霍巴汀对钠(V)通道的影响

Pérez, Rebeca; Figueredo, Claudia; Burgos, Viviana; Cabrera-Pardo, Jaime R; Schmidt, Bernd; Heydenreich, Matthias; Koch, Andreas; Deuis, Jennifer R; Vetter, Irina; Paz, Cristian