日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimizing uPAR-targeting radiopeptides for improved tissue distribution: progress towards radionuclide therapy

优化靶向 uPAR 的放射性肽以改善组织分布:放射性核素治疗的进展

Vaccarin, Christian; Beyer, Darja; Schmid, Jerome V; Klein, Bastian; Jegathasan, Jathursa; Behera, Shreshtha; Deupi, Xavier; Schibli, Roger; Müller, Cristina

Cyclic peptide inhibitors function as molecular glues to stabilize Gq/11 heterotrimers

环肽抑制剂起到分子胶的作用,稳定Gq/11异源三聚体。

Mühle, Jonas; Alenfelder, Judith; Rodrigues, Matthew J; Jürgenliemke, Lars; Guixà-González, Ramon; Grätz, Lukas; Andres, Fabio; Bacchin, Arianna; Hennig, Michael; Schihada, Hannes; Crüsemann, Max; König, Gabriele M; Schertler, Gebhard; Kostenis, Evi; Deupi, Xavier

Coral anthozoan-specific opsins employ a novel chloride counterion for spectral tuning

珊瑚虫特有的视蛋白利用一种新型的氯离子反离子进行光谱调谐。

Sakai, Yusuke; Sen, Saumik; Sugihara, Tomohiro; Kakeyama, Yukiya; Iwasaki, Makoto; Schertler, Gebhard F X; Deupi, Xavier; Koyanagi, Mitsumasa; Terakita, Akihisa

Design and Preclinical Evaluation of Novel uPAR-Targeting Radiopeptides Modified with an Albumin-Binding Entity

利用白蛋白结合实体修饰的新型uPAR靶向放射性肽的设计和临床前评估

Beyer, Darja; Vaccarin, Christian; Schmid, Jerome V; Deberle, Luisa M; Deupi, Xavier; Schibli, Roger; Müller, Cristina

Active state structures of a bistable visual opsin bound to G proteins

与G蛋白结合的双稳态视蛋白的活性状态结构

Tejero, Oliver; Pamula, Filip; Koyanagi, Mitsumasa; Nagata, Takashi; Afanasyev, Pavel; Das, Ishita; Deupi, Xavier; Sheves, Mordechai; Terakita, Akihisa; Schertler, Gebhard F X; Rodrigues, Matthew J; Tsai, Ching-Ju

Calcineurin-fusion facilitates cryo-EM structure determination of a Family A GPCR.

钙调磷酸酶融合促进了A家族GPCR的冷冻电镜结构测定

Xu Jun, Chen Geng, Wang Haoqing, Cao Sheng, Heng Jie, Deupi Xavier, Du Yang, Kobilka Brian K

Development of radiofluorinated MLN-4760 derivatives for PET imaging of the SARS-CoV-2 entry receptor ACE2

开发用于SARS-CoV-2进入受体ACE2 PET成像的放射性氟化MLN-4760衍生物

Wang, Jinling; Beyer, Darja; Vaccarin, Christian; He, Yingfang; Tanriver, Matthias; Benoit, Roger; Deupi, Xavier; Mu, Linjing; Bode, Jeffrey W; Schibli, Roger; Müller, Cristina

Study of Photoselectivity in Linear Conjugated Chromophores Using the XMS-CASPT2 Method

利用XMS-CASPT2方法研究线性共轭发色团的光选择性

Sen, Saumik; Deupi, Xavier

Structural Elements Directing G Proteins and β-Arrestin Interactions with the Human Melatonin Type 2 Receptor Revealed by Natural Variants

天然变异体揭示了指导 G 蛋白和 β-arrestin 与人类褪黑素 2 型受体相互作用的结构元件

Plouffe, Bianca; Karamitri, Angeliki; Flock, Tilman; Gallion, Jonathan M; Houston, Shane; Daly, Carole A; Bonnefond, Amélie; Guillaume, Jean-Luc; Le Gouill, Christian; Froguel, Phillipe; Lichtarge, Olivier; Deupi, Xavier; Jockers, Ralf; Bouvier, Michel

High-mass MALDI-MS unravels ligand-mediated G protein-coupling selectivity to GPCRs

高通量MALDI-MS揭示配体介导的G蛋白偶联对GPCR的选择性

Wu, Na; Olechwier, Agnieszka M; Brunner, Cyrill; Edwards, Patricia C; Tsai, Ching-Ju; Tate, Christopher G; Schertler, Gebhard F X; Schneider, Gisbert; Deupi, Xavier; Zenobi, Renato; Ma, Pikyee