日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Solid-phase peptide head-to-side chain cyclodimerization: discovery of C(2)-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

固相肽头链侧链环化二聚化:发现对人类黑素皮质素受体具有强效活性的 C(2)-对称环内酰胺杂化 α-黑素细胞刺激激素 (MSH)/刺豚鼠信号蛋白 (ASIP) 类似物

Alexander V Mayorov, Minying Cai, Erin S Palmer, Zhihua Liu, James P Cain, Josef Vagner, Dev Trivedi, Victor J Hruby

Opioid and melanocortin receptors: do they have overlapping pharmacophores?

阿片类药物和黑皮质素受体:它们是否具有重叠的药效团?

Yeon Sun Lee, Richard S Agnes, James P Cain, Vinod Kulkarni, Minying Cai, Christine Salibay, Kathy Ciano, Ravil Petrov, Alexander Mayorov, Josef Vagner, Dev Trivedi, Peg Davis, Shou-wu Ma, Josephine Lai, Frank Porreca, Ruben Vardanyan, Victor J Hruby

Effects of macrocycle size and rigidity on melanocortin receptor-1 and -5 selectivity in cyclic lactam alpha-melanocyte-stimulating hormone analogs

大环大小和刚性对环内酰胺 α-促黑素细胞激素类似物中黑皮质素受体-1 和 -5 选择性的影响

Alexander V Mayorov, So-Yeop Han, Minying Cai, Matthew R Hammer, Dev Trivedi, Victor J Hruby