日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells

强效且选择性的 SETDB1 共价负变构调节剂可降低细胞中的甲基转移酶活性

Mélanie Uguen, Devan J Shell, Madhushika Silva, Yu Deng, Fengling Li, Magdalena M Szewczyk, Ka Yang, Yani Zhao, Michael A Stashko, Jacqueline L Norris-Drouin, Jarod M Waybright, Serap Beldar, Justin M Rectenwald, Angie L Mordant, Thomas S Webb, Laura E Herring, Cheryl H Arrowsmith, Suzanne Ackloo, S

Barriers and Facilitators to Video Telehealth Use in Low-Income Hispanic Patients: A Theory of Planned Behavior Perspective

低收入西班牙裔患者使用视频远程医疗的障碍和促进因素:基于计划行为理论的视角

Peterson, Devan J; de Haro, Cristina M; Kilgore, David B; Sorkin, Dara H; Gago-Masague, Sergio; Billimek, John

Expansion of DNA-Encoded Library Hits Using Generative Chemistry and Ultra-Large Compound Catalogs

利用生成化学和超大型化合物目录扩展DNA编码化合物库

Novy, Brandon; Lin, Shu-Hang; Shell, Devan J; Maxfield, Travis; Merten, Eric M; Wellnitz, James; Guduru, Shiva K R; Hardy, P Brian; Pearce, Kenneth H; Popov, Konstantin I

Identification of Covalent Cyclic Peptide Inhibitors in mRNA Display

mRNA展示技术中共价环肽抑制剂的鉴定

Iskandar, Sabrina E; Chiou, Lilly F; Leisner, Tina M; Shell, Devan J; Norris-Drouin, Jacqueline L; Vaziri, Cyrus; Pearce, Kenneth H; Bowers, Albert A

Discovery of a 53BP1 Small Molecule Antagonist Using a Focused DNA-Encoded Library Screen

利用聚焦DNA编码文库筛选发现53BP1小分子拮抗剂

Devan J Shell ,Caroline A Foley ,Qinhong Wang ,Chelsea M Smith ,Shiva K R Guduru ,Hong Zeng ,Aiping Dong ,Jacqueline L Norris-Drouin ,Matthew Axtman ,P Brian Hardy ,Gaorav Gupta ,Levon Halabelian ,Stephen V Frye ,Lindsey I James ,Kenneth H Pearce

SETDB1 Triple Tudor Domain Ligand, (R, R)-59, Promotes Methylation of Akt1 in Cells

SETDB1 三重 Tudor 结构域配体 (R, R)-59 促进细胞中 Akt1 甲基化

Mélanie Uguen, Yu Deng, Fengling Li, Devan J Shell, Jacqueline L Norris-Drouin, Michael A Stashko, Suzanne Ackloo, Cheryl H Arrowsmith, Lindsey I James, Pengda Liu, Kenneth H Pearce, Stephen V Frye

Identifying drivers of breast cancer metastasis in progressively invasive subpopulations of zebrafish-xenografted MDA-MB-231

识别斑马鱼异种移植 MDA-MB-231 的渐进性侵袭性亚群中乳腺癌转移的驱动因素

Jerry Xiao, Joseph R McGill, Apsra Nasir, Alexander Lekan, Bailey Johnson, Devan J Wilkins, Gray W Pearson, Kandice Tanner, Hani Goodarzi, Eric Glasgow, Richard Schlegel, Seema Agarwal

A multiplex preclinical model for adenoid cystic carcinoma of the salivary gland identifies regorafenib as a potential therapeutic drug

涎腺腺样囊性癌的多重临床前模型确定瑞戈非尼是一种潜在的治疗药物

Chen Chen, Sujata Choudhury, Darawalee Wangsa, Chamille J Lescott, Devan J Wilkins, Praathibha Sripadhan, Xuefeng Liu, Danny Wangsa, Thomas Ried, Christopher Moskaluk, Michael J Wick, Eric Glasgow, Richard Schlegel, Seema Agarwal