Combined inhibition of MAP kinase and KIT signaling synergistically destabilizes ETV1 and suppresses GIST tumor growth
MAP 激酶和 KIT 信号传导的联合抑制可协同破坏 ETV1 的稳定性并抑制 GIST 肿瘤的生长
期刊:Cancer Discovery
影响因子:29.7
doi:10.1158/2159-8290.CD-14-0985
Leili Ran, Inna Sirota, Zhen Cao, Devan Murphy, Yuedan Chen, Shipra Shukla, Yuanyuan Xie, Michael C Kaufmann, Dong Gao, Sinan Zhu, Ferdinando Rossi, John Wongvipat, Takahiro Taguchi, William D Tap, Ingo K Mellinghoff, Peter Besmer, Cristina R Antonescu, Yu Chen, Ping Chi