日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Arylsulfonamide KCN1 inhibits in vivo glioma growth and interferes with HIF signaling by disrupting HIF-1α interaction with cofactors p300/CBP.

芳基磺酰胺 KCN1 可抑制体内神经胶质瘤的生长,并通过破坏 HIF-1α 与辅助因子 p300/CBP 的相互作用来干扰 HIF 信号传导

Yin Shaoman, Kaluz Stefan, Devi Narra S, Jabbar Adnan A, de Noronha Rita G, Mun Jiyoung, Zhang Zhaobin, Boreddy Purushotham R, Wang Wei, Wang Zhibo, Abbruscato Thomas, Chen Zhengjia, Olson Jeffrey J, Zhang Ruiwen, Goodman Mark M, Nicolaou K C, Van Meir Erwin G

Design and synthesis of novel small-molecule inhibitors of the hypoxia inducible factor pathway

设计并合成新型缺氧诱导因子通路小分子抑制剂

Mooring, Suazette Reid; Jin, Hui; Devi, Narra S; Jabbar, Adnan A; Kaluz, Stefan; Liu, Yuan; Van Meir, Erwin G; Wang, Binghe

Sulfonamides as a new scaffold for hypoxia inducible factor pathway inhibitors

磺胺类药物作为缺氧诱导因子通路抑制剂的新型支架

Tan, Chalet; de Noronha, Rita G; Devi, Narra S; Jabbar, Adnan A; Kaluz, Stefan; Liu, Yuan; Mooring, Suazette Reid; Nicolaou, K C; Wang, Binghe; Van Meir, Erwin G

Vasculostatin inhibits intracranial glioma growth and negatively regulates in vivo angiogenesis through a CD36-dependent mechanism

血管抑素通过CD36依赖性机制抑制颅内胶质瘤生长并负向调控体内血管生成。

Kaur, Balveen; Cork, Sarah M; Sandberg, Eric M; Devi, Narra S; Zhang, Zhaobin; Klenotic, Philip A; Febbraio, Maria; Shim, Hyunsuk; Mao, Hui; Tucker-Burden, Carol; Silverstein, Roy L; Brat, Daniel J; Olson, Jeffrey J; Van Meir, Erwin G