日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Coronavirus Main Protease Inhibitors with Enhanced Brain Exposure and Potent Oral Efficacy in SARS-CoV-2 and MERS Infection Models

在SARS-CoV-2和MERS感染模型中发现具有增强脑暴露和强效口服疗效的冠状病毒主要蛋白酶抑制剂

Lizzadro, Luca; Li, Jiapeng; Taha, Taha Y; Degotte, Gilles; Detomasi, Tyler C; Zapatero-Belinchon, Francisco J; Hantz, Eric R; Huang, Sijie; Matsui, Yusuke; Henderson, Will R; McCann, Jack T; Montano, Mauricio; Rosecrans, Julia; Torres Pomares, Daniel F; McGovern, Briana L; Diaz-Tapia, Randy; Benjamin, Jared; Gordon, Mary E; Suazo, Isidora D; Settineri, Nicholas S; Diallo, Amy; Krogan, Nevan J; Shoichet, Brian K; Verba, Kliment A; Albrecht, Randy; García-Sastre, Adolfo; White, Kris M; Ott, Melanie; Craik, Charles S; Renslo, Adam R

Linking biochemical and cellular efficacy of MERS coronavirus main protease inhibitors

关联MERS冠状病毒主蛋白酶抑制剂的生化和细胞功效

La, Van N T; Lahav, Noa; Rodriguez, Mario; Diaz-Tapia, Randy; McGovern, Briana; Benjamin, Jared; Barr, Haim; White, Kris M; Kang, Lulu; Chodera, John D; Minh, David D L

Structure-Activity Relationship Studies Towards Analogues of Pleconaril as Novel Enterovirus-D68 Capsid-Targeting Antivirals

针对新型肠道病毒D68衣壳靶向抗病毒药物的普利可那利类似物的结构-活性关系研究

Cousins, David L; Griffen, Ed J; Stacey, Jessica; Lee, Alpha A; Filimonova, Yuliia; Hlavin, Anton; Holota, Yuliia; Khmil, Roman; Kordubailo, Mykyta; Kostinov, Oleksii; Lesyk, Dmytro; Logvinenko, Ivan; Lototska, Mariia; Lysenko, Viacheslav; Pashchenko, Anna; Pavlichenko, Mariia; Rodnichenko, Anzhela; Tkachenko, Anton; Hurst, Brett L; Julander, Justin G; Wang, Hong; Pearl, Rebecca; Benjamin, Jared; Diaz-Tapia, Randy; Gordon, Mary E; Albrecht, Randy A; White, Kris

Adaptive multi-epitope targeting and avidity-enhanced nanobody platform for ultrapotent, durable antiviral therapy.

用于超强效、持久抗病毒治疗的自适应多表位靶向和亲和力增强纳米抗体平台

Xiang Yufei, Xu Jialu, McGovern Briana L, Ranzenigo Anna, Huang Wei, Sang Zhe, Shen Juan, Diaz-Tapia Randy, Pham Ngoc Dung, Teunissen Abraham J P, Rodriguez M Luis, Benjamin Jared, Taylor Derek J, van Leent Mandy M T, White Kris M, García-Sastre Adolfo, Zhang Peijun, Shi Yi