日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

RNA-targeted proteomics identifies YBX1 as critical for efficient HCMV mRNA translation.

RNA靶向蛋白质组学鉴定出YBX1对于HCMV mRNA的有效翻译至关重要

Dickmander Rebekah J, Lenarcic Erik M, Sears John D, Hale Andrew E, Moorman Nathaniel J

Novel Computational Pipeline to Identify Target Sites for Broad Spectrum Antiviral Drugs

用于识别广谱抗病毒药物靶点的新型计算流程

Sears, John D; Popov, Konstantin I; Sylvester, Paul; Dickmander, Rebekah; Loome-Diaz, Jennifer; Chang, Che-Kang; Huff, Julia; Sanders, Wes; Saba, Nicholas A; Sorensen, Madeleine; Drobish, Adam M; May, Nicholas A; Namitz, Kevin; Fecko, Julia; Arnold, Jamie J; Yennawar, Neela H; Cameron, Craig E; Morrison, Thomas E; Tropsha, Alexander; Heise, Mark T; Moorman, Nathaniel J

Lethal COVID-19 associates with RAAS-induced inflammation for multiple organ damage including mediastinal lymph nodes

致命的 COVID-19 与 RAAS 诱导的炎症有关,可导致包括纵隔淋巴结在内的多器官损伤。

Topper, Michael J; Guarnieri, Joseph W; Haltom, Jeffrey A; Chadburn, Amy; Cope, Henry; Frere, Justin; An, Julia; Borczuk, Alain; Sinha, Saloni; Kim, JangKeun; Park, Jiwoon; Butler, Daniel; Meydan, Cem; Foox, Jonathan; Bram, Yaron; Richard, Stephanie A; Epsi, Nusrat J; Agan, Brian; Chenoweth, Josh G; Simons, Mark P; Tribble, David; Burgess, Timothy; Dalgard, Clifton; Heise, Mark T; Moorman, Nathaniel J; Baxter, Victoria K; Madden, Emily A; Taft-Benz, Sharon A; Anderson, Elizabeth J; Sanders, Wes A; Dickmander, Rebekah J; Beigel, Katherine; Widjaja, Gabrielle A; Janssen, Kevin A; Lie, Timothy; Murdock, Deborah G; Angelin, Alessia; Soto Albrecht, Yentli E; Olali, Arnold Z; Cen, Zimu; Dybas, Joseph; Priebe, Waldemar; Emmett, Mark R; Best, Sonja M; Kelsey Johnson, Maya; Trovao, Nidia S; Clark, Kevin B; Zaksas, Victoria; Meller, Robert; Grabham, Peter; Schisler, Jonathan C; Moraes-Vieira, Pedro M; Pollett, Simon; Mason, Christopher E; Syrkin Wurtele, Eve; Taylor, Deanne; Schwartz, Robert E; Beheshti, Afshin; Wallace, Douglas C; Baylin, Stephen B

More than an Amide Bioisostere: Discovery of 1,2,4-Triazole-containing Pyrazolo[1,5- a]pyrimidine Host CSNK2 Inhibitors for Combatting β-Coronavirus Replication

不仅仅是酰胺生物电子等排体:发现含 1,2,4-三唑的吡唑并[1,5- a]嘧啶宿主 CSNK2 抑制剂用于对抗 β-冠状病毒复制

Han Wee Ong, Xuan Yang, Jeffery L Smith, Rebekah J Dickmander, Jason W Brown, Tammy M Havener, Sharon Taft-Benz, Stefanie Howell, Marcia K Sanders, Jacob L Capener, Rafael M Couñago, Edcon Chang, Andreas Krämer, Nathaniel J Moorman, Mark Heise, Alison D Axtman, David H Drewry, Timothy M Willson

Specific RNA structures in the 5' untranslated region of the human cytomegalovirus major immediate early transcript are critical for efficient virus replication

人类巨细胞病毒主要立即早期转录本 5’ 非翻译区中的特定 RNA 结构对于病毒的有效复制至关重要

Bekah Dickmander, Andrew Hale, Wes Sanders, Erik Lenarcic, Ben Ziehr, Nathaniel J Moorman

Strategic Fluorination to Achieve a Potent, Selective, Metabolically Stable, and Orally Bioavailable Inhibitor of CSNK2

通过战略性氟化获得强效、选择性、代谢稳定且口服生物可利用的 CSNK2 抑制剂

Han Wee Ong, Xuan Yang, Jeffery L Smith, Sharon Taft-Benz, Stefanie Howell, Rebekah J Dickmander, Tammy M Havener, Marcia K Sanders, Jason W Brown, Rafael M Couñago, Edcon Chang, Andreas Krämer, Nathaniel J Moorman, Mark Heise, Alison D Axtman, David H Drewry, Timothy M Willson

Protein phosphatase 1 suppresses PKR/EIF2α signaling during human cytomegalovirus infection

蛋白磷酸酶1在人巨细胞病毒感染期间抑制PKR/EIF2α信号传导

Lenarcic, Erik M; Hale, Andrew E; Vincent, Heather A; Dickmander, Rebekah J; Sanders, Wes; Moorman, Nathaniel J

Identification of 4-(6-((2-methoxyphenyl)amino)pyrazin-2-yl)benzoic acids as CSNK2A inhibitors with antiviral activity and improved selectivity over PIM3

鉴定出 4-(6-((2-甲氧基苯基)氨基)吡嗪-2-基)苯甲酸类化合物为 CSNK2A 抑制剂,具有抗病毒活性,且选择性优于 PIM3。

Galal, Kareem A; Krämer, Andreas; Strickland, Benjamin G; Smith, Jeffery L; Dickmander, Rebekah J; Moorman, Nathaniel J; Willson, Timothy M

Optimization of 3-Cyano-7-cyclopropylamino-pyrazolo[1,5- a]pyrimidines toward the Development of an In Vivo Chemical Probe for CSNK2A

优化 3-氰基-7-环丙基氨基-吡唑并[1,5- a]嘧啶以开发 CSNK2A 体内化学探针

Xuan Yang, Han Wee Ong, Rebekah J Dickmander, Jeffery L Smith, Jason W Brown, William Tao, Edcon Chang, Nathaniel J Moorman, Alison D Axtman, Timothy M Willson

Vandetanib Blocks the Cytokine Storm in SARS-CoV-2-Infected Mice

凡德他尼阻断 SARS-CoV-2 感染小鼠的细胞因子风暴

Ana C Puhl, Giovanni F Gomes, Samara Damasceno, Ethan J Fritch, James A Levi, Nicole J Johnson, Frank Scholle, Lakshmanane Premkumar, Brett L Hurst, Felipe Lee-Montiel, Flavio P Veras, Sabrina S Batah, Alexandre T Fabro, Nathaniel J Moorman, Boyd L Yount, Rebekah J Dickmander, Ralph S Baric, Kenneth