Identification of a Highly Cooperative PROTAC Degrader Targeting GTP-Loaded KRAS(On) Alleles
鉴定一种高度协同的PROTAC降解酶,该酶靶向GTP结合的KRAS(On)等位基因
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.5c10354
Vetma, Vesna; Puoti, Ilaria; Karolak, Natalia K; Chakraborti, Sohini; Diers, Emelyne; Girardi, Enrico; Khan, Shakil; Kidd, Giorgia; Kropatsch, Katrin G; Mclennan, Ross; O'Connor, Suzanne; Samwer, Matthias; Trainor, Nicole; Whitworth, Claire; Wijaya, Andre J; Wong, Jeff Y F; Zollman, David; Farnaby, William; Popow, Johannes; Ciulli, Alessio; Ettmayer, Peter; McAulay, Kirsten