Peptidomimetic Phenoxymethyl Ketone Warheads as Potent Dual-Mode Inhibitors against SARS-CoV-2 M(pro) and Cathepsin
肽模拟苯氧甲基酮弹头作为强效双模式抑制剂,可抑制SARS-CoV-2 M(pro)和组织蛋白酶
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c03147
Porzberg, Miriam R B; Groenewold, G J Mirjam; Lyoo, Heyrhyoung; Jakob, Alexander K M H; Titulaer, Willem H C; Cavina, Lorenzo; Poelaert, Katrien C K; Zwaagstra, Marleen; Dieteren, Cindy E J; Lemmers, Jaap G H; Hamdani, S Hakim; van Buuren, Bernd N M; Ackerschott, Bart; Platteeuw, Johannes; Michorius, Joey; Martina, Byron E E; Feiters, Martin C; Gironés, Daniel; van Kuppeveld, Frank J M; van Hemert, Martijn J; Rutjes, Floris P J T