日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological and structural characterization of vibostolimab, a novel anti-TIGIT blocking antibody for cancer immunotherapy

对新型抗TIGIT阻断抗体vibostolimab进行药理学和结构表征,该抗体可用于癌症免疫治疗。

Thierry O Fischmann ,Daniel Malashock ,Eunseon Ahn ,Hongmei Wang ,Komal Pradhan ,Jeffery Grein ,Srishti Chakravorty ,Soheila Bahmanjah ,David Ban ,Ellen Chien ,Mark Hsieh ,Todd Mayhood ,Jing Yuan ,Janica C Wong ,Maribel Beaumont ,Jeanne Baker ,Mark A McCoy ,Mingmei Cai ,Douglas Wilson ,Wendy Blumenschein ,Sybil M G Williams ,Laurence Fayadat-Dilman ,Wolfgang Seghezzi ,Tanya Keenan ,Jin-Hwan Han

Unlocking the reactivity of the C-In bond: alkyl indium reagents as a source of radicals under photocatalytic conditions

释放C-In键的反应活性:烷基铟试剂作为光催化条件下自由基的来源

Gladkov, Anton A; Levin, Vitalij V; Cheboksarov, Demian Y; Dilman, Alexander D

Biologics developability data analysis using hierarchical clustering accelerates candidate lead selection, optimization, and preformulation screening.

利用层次聚类进行生物制剂可开发性数据分析,可以加速候选先导化合物的选择、优化和制剂前筛选

Metcalf Kevin James, Wo Galen, Zaragoza Jan Paulo, Raoufi Fahimeh, Baker Jeanne, Chen Daoyang, Derebe Mehabaw, Hogan Jason, Hsu Amy, Kofman Esther, Leigh David, Li Mandy, Malashock Dan, Mann Cate, Motlagh Soha, Park Jihea, Sathiyamoorthy Karthik, Shidhore Madhura, Tang Yinyan, Teng Kevin, Williams Katharine, Waight Andrew, Yilmaz Sultan, Zhang Fan, Zhong Huimin, Fayadat-Dilman Laurence, Bailly Marc

Structural Characterization of Linker Shielding in ADC Site-Specific Conjugates

ADC位点特异性偶联物中连接基团屏蔽的结构表征

Jaime-Garza, Maru; Waight, Andrew; Hudlikar, Manish; Eddins, Michael J; Rasti, Elnaz S; Zaragoza, Jan Paulo T; Fayadat-Dilman, Laurence; Chrencik, Jill E; Gabelli, Sandra B; Chen, Yun-Ting; Noland, Cameron L

Characterizing Monoclonal Antibody Aggregation Using Charge Detection Mass Spectrometry and Industry Standard Methods

利用电荷检测质谱和行业标准方法表征单克隆抗体聚集

Jordan, Jacob S; Harper, Conner C; Zhang, Fan; Kofman, Esther; Sam, Miranda; Zaragoza, Jan Paulo; Bhagwat, Bhagyashree; Fayadat-Dilman, Laurence; Williams, Evan R

Charge Detection Mass Spectrometry Reveals Conformational Heterogeneity in Megadalton-Sized Monoclonal Antibody Aggregates

电荷检测质谱揭示兆道尔顿级单克隆抗体聚集体的构象异质性

Jordan, Jacob S; Harper, Conner C; Zhang, Fan; Kofman, Esther; Li, Mandy; Sathiyamoorthy, Karthik; Zaragoza, Jan Paulo; Fayadat-Dilman, Laurence; Williams, Evan R

Direct conversion of carboxylic acids to free thiols via radical relay acridine photocatalysis enabled by N-O bond cleavage

通过NO键断裂实现的自由基接力吖啶光催化,将羧酸直接转化为游离硫醇

Lipilin, Dmitry L; Zubkov, Mikhail O; Kosobokov, Mikhail D; Dilman, Alexander D

Exploring the use of COVID-19 antigen rapid diagnostic tests among displaced populations in Iraq: findings from a pilot project in four IDP camps

探索在伊拉克流离失所人群中使用新冠病毒抗原快速诊断测试:来自四个境内流离失所者营地的试点项目的研究结果

Ammar, Lara Abou; Wolfe, Caitlin M; Nagib, Lamiaa; Slebei, Mohammed; Shawkat, Sezan; Amo, Dilman; Abdullah, Raveen; Abdulmalik, Rawshan; Amin, Hiwa Muhammed; Shafiq, Huda; Hafthalah, Shivan; Qahraman, Aso; Mohammed, Jirjees; Ghawji, Hassan; Satyanarayana, Srinath; Wilson, Nevin; Sarin, Sanjay; Kao, Kekeletso; Ghusayni, Nellie

Understanding the Landscape: The Emergence of Artificial Intelligence (AI), ChatGPT, and Google Bard in Gastroenterology

了解现状:人工智能 (AI)、ChatGPT 和 Google Bard 在胃肠病学领域的兴起

Rammohan, Rajmohan; Joy, Melvin V; Magam, Sai Greeshma; Natt, Dilman; Magam, Sai Reshma; Pannikodu, Leeza; Desai, Jiten; Akande, Olawale; Bunting, Susan; Yost, Robert M; Mustacchia, Paul

Addressing the Gap: Racial Disparities and Public Health Strategies in the Epidemiology of Gastrointestinal Stromal Tumors

弥合差距:胃肠道间质瘤流行病学中的种族差异和公共卫生策略

Rammohan, Rajmohan; Joy, Melvin; Magam, Sai Greeshma; Lau, Wing Hang; Natt, Dilman; Tadikonda, Abhishek; Magam, Sai Reshma; Pannikodu, Leeza; Desai, Jiten; Jiyani, Rucha; Sheikh, Saher; Gomez, Sandra; Bunting, Susan; Anand, Prachi; Subramani, Krishnaiyer; Mustacchia, Paul